T8409SYN1143c-Met/HGFR,SYN-1143,tumor,RON,dual,inhibit,SYN1143,SYN 1143,cancer,Inhibitor,c-Met

AMG-1 is a potent inhibitor of human RON and c-Met.In vitro kinase assays showed that compound I is a potent inhibitor of human RON and c-Met with IC50s of 9 and 4 nmol/L, respectively.

价 格：￥电议型 号：T8409产 地：中国大陆

T9816ArofyllineLAS-31025,inhibit,Arofylline,LAS31025,Phosphodiesterase (PDE),Inhibitor

Arofylline is a PDE4 inhibitor and can be used for asthma studies.

价 格：￥电议型 号：T9816产 地：中国大陆

T7395LanifibranorInhibitor,IVA 337,Lanifibranor,inhibit,PPAR,Peroxisome proliferator-activated receptors,

Lanifibranor is an agonist of peroxisome proliferator-activated receptors (PPARs) with EC50 values of 1,537, 866, and 206 nM for human recombinant PPARα, PPARβ, and PPARγ, respectively, for transactivation activity

价 格：￥电议型 号：T7395产 地：中国大陆

T7486Imeglimin hydrochlorideEMD387008,inhibit,mitochondrial,lowering,insulin,Mitochondrial Metabolism,ora

Imeglimin hydrochloride prevents human endothelial cell death by inhibiting mitochondrial permeability transition without inhibiting mitochondrial respiration.

价 格：￥电议型 号：T7486产 地：中国大陆

T35973Cholesterol-5α,6α-epoxide

Cholesterol-5α,6α-epoxide is the metabolite of cholesterol produced by oxidation. Cholesterol-5α,6α-epoxide induces triacylglycerol biosynthesis by binding to LXRβ following tamoxifen and PBPE application.

价 格：￥电议型 号：T35973产 地：中国大陆

T9115Vanillic AcidNuclear factor-κB,Vanillic Acid,NF-κB,inhibit,Bacterial,Nuclear factor-kappaB,Endogenou

Vanillic acid is used as a condiment in food,which used in wine and vinegar. It is an intermediate in the production of vanillin from ferulic acid.

价 格：￥电议型 号：T9115产 地：中国大陆

T60075Thieno[2,3-b]pyridine-2-carboxamide, 3-amino-N-[5-[4-(2,3-dichlorophenyl)-1-piperazinyl]pentyl]-4,6-

Thieno[2,3-b]pyridine-2-carboxamide, 3-amino-N-[5-[4-(2,3-dichlorophenyl)-1-piperazinyl]pentyl]-4,6-dimethyl- is a ligand targeting the dopamine D2 receptor.

价 格：￥电议型 号：T60075产 地：中国大陆

T9121AG-636inhibit,oral,AG 636,AG-636,reversible,DHODH,anticancer,AG636,Inhibitor,Dihydroorotate Dehydrog

AG-636 is a potent, reversible, selective and orally active DHODH inhibitor(IC50 of 17 nM). It has strong anticancer effects.

价 格：￥电议型 号：T9121产 地：中国大陆

T37445EtanerceptEtanercept

Etanercept, a dimeric fusion protein that binds TNF, acts as a TNF inhibitor. Etanercept competitively inhibits the binding of both TNF-α and TNF-β to cell surface TNF receptors, rendering TNF biologically inactive. Etanercept shows efficacy against rheumatoid arthritis, juvenile idiopathic arthritis, and plaque psoriasis.

价 格：￥电议型 号：T37445产 地：中国大陆

T8507MAC-545496Bacterial,S. aureus,Antivirulence,Inhibitor,MAC545496,mprF,nanomolar,GraR,MAC-545496,MRSA,

MAC-545496 is a glycopeptide-resistance-associated protein R (GraR) inhibitor, is an antivirulence agent.

价 格：￥电议型 号：T8507产 地：中国大陆

T7222GS-441524GS-441524,Inhibitor,feline,SARS coronavirus,virus,FIPV,infectious,peritonitis,DNA/RNA Synth

GS-441524 treatment of cats with naturally occurring feline infectious peritonitis.

价 格：￥电议型 号：T7222产 地：中国大陆

T5903Sitagliptin Intermediate 2Sitagliptin Intermediate 2

价 格：￥电议型 号：T5903产 地：中国大陆

TN1490Chrysoeriolinhibit,Endogenous Metabolite,Inhibitor,Chrysoeriol

Chrysoeriol has antioxidant, antiinflammatory, antitumor, antimicrobial, antiviral, and free radical scavenging activities, it also shows selective bronchodilator effect.

价 格：￥电议型 号：TN1490产 地：中国大陆

T6S1894LinderaneCYPs,Cytochrome P450,Linderane,inhibit,Inhibitor

1. Linderane was characterized as a mechanism-based inactivator of CYP2C9.

价 格：￥电议型 号：T6S1894产 地：中国大陆

T60028MM41inhibit,G-quadruplex,MM41,MM 41,PaCa-2,pancreatic cancer,A549,Inhibitor,cancer,stabilizer,RCC4,7

MM41 is a human telomeric and gene promoter DNA quadruplex stabilizer with an IC50 of <10 nM against the MIA PaCa-2 pancreatic cancer cell line.

价 格：￥电议型 号：T60028产 地：中国大陆

T8930CID44216842diseases,neutrophils,ovarian,disorders,Cdc42,fibroblasts,breast,hepatitis C,CID 44216842,

CID44216842 is a potent Cdc42-selective guanine nucleotide binding lead inhibitor. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 1.0 and 1.2 μM in GTP binding assay, respectively. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 0.3 and 0.5 μM in GDP binding assay, respectively. Use as a molecular probe.

价 格：￥电议型 号：T8930产 地：中国大陆

T7546BethoxazinBethoxazin,inhibit,Inhibitor,Bacterial

Bethoxazin is a new broad spectrum industrial microbicide.

价 格：￥电议型 号：T7546产 地：中国大陆

T9349IXA4endoplasmic reticulum (ER) proteostasis,UPR,protein secretion,Inhibitor,Inositol requiring enzym

IXA4 is a highly selective, nontoxic activator of IRE1/XBP1s and reduces APP secretion by activating IRE1. IXA4-stimulated IRE1 activation also enhanced pancreatic function.

价 格：￥电议型 号：T9349产 地：中国大陆

T16845Sarolanerdog,Sarolaner,Parasite,PF 6450567,flea,Inhibitor,oral,inhibit,isoxazoline,tick,PF6450567

Sarolaner is an orally active and broad-spectrum ectoparasiticide (LC80: 0.3 μg/mL against C. felis and an LC100: 0.003 μg/mL against O. turicata).

价 格：￥电议型 号：T16845产 地：中国大陆

TN6848Piperonylic acidformation,virus,natural,inactivator,Cytochrome P450,Piperonylic acid,quasi-irreversi

Piperonylic acid is a natural molecule bearing a methylenedioxy function that closely mimics the structure of trans-cinnamic acid. Piperonylic acid selectively inactivate the CYP73A P450 subpopulation.

价 格：￥电议型 号：TN6848产 地：中国大陆