T37082HS271HS271,HS-271

HS271 is a selective, highly potent and orally active IRAK4 inhibitor (IC50= 7.2 μM). HS271 shows excellent enzymatic and cellular activities, as well as excellent pharmacokinetic properties.

价 格：￥电议型 号：T37082产 地：中国大陆

TQ0271Falnidamol

Falnidamol is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. Falnidamol displays > 1000-fold lower potency against ErbB2 (IC50=3.4 μM) and a range of other related tyrosine kinases (IC50>10 μM). Falnidamol is a pyrimido-pyrimidine compound and has anti-cancer activity.

价 格：￥电议型 号：TQ0271产 地：中国大陆

T6644RolipramHuman immunodeficiency virus,SB95952,Rolipram,ZK62711,Inhibitor,SB-95952,Bacterial,Phosphodi

Rolipram is a phosphodiesterase 4 inhibitor with antidepressant properties.

价 格：￥电议型 号：T6644产 地：中国大陆

TPL0053Compound 227105-11-5Compound 227105 11 5,Compound 227105115

价 格：￥电议型 号：TPL0053产 地：中国大陆

T7946AER-271Inhibitor,AER-271,AQP4,AER-270,stroke,inhibit,aquaporin-4,injury,AER 271,acute,AER271,CNS,isc

AER-271 is an inhibitor of aquaporin-4.

价 格：￥电议型 号：T7946产 地：中国大陆

T9271RAD51-IN-1cancer,inhibit,tumor cell,chemotherapy,RAD51 IN 1,Inhibitor,RAD51,DNA damage,RAD-51-IN-1,R

Rad51-in-1 is a derivative of B02 and an effective inhibitor of Rad51.

价 格：￥电议型 号：T9271产 地：中国大陆

T38271TH1217

TH1217 is a potent and selective dCTPase pyrophosphatase 1 (dCTPase) inhibitor, with an IC50 of 47 nM. TH1217 enhances the cytotoxic effect of cytidine analogues in leukemia cells. TH1217 also could modulate SARS-Cov-2 interactors, so it shows activity of against COVID-19.

价 格：￥电议型 号：T38271产 地：中国大陆

T827110Z-Nonadecenoic acid10Z Nonadecenoic acid,Endogenous Metabolite,Inhibitor,inhibit,10Z-Nonadecenoic

10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.

价 格：￥电议型 号：T8271产 地：中国大陆

TN1271Scutellarein tetramethyl etherBacterial,Inhibitor,inhibit,Scutellarein tetramethyl ether

Scutellarein tetramethyl ether is extracted from Siam weeds and exhibits anti-inflammatory activity through NF-κB pathway.

价 格：￥电议型 号：TN1271产 地：中国大陆

TP1271LCalmodulin-Dependent Protein Kinase II 290-309 acetateCalmodulin Dependent Protein Kinase II 290 309

Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).

价 格：￥电议型 号：TP1271L产 地：中国大陆

T9846WAY-327157WAY327157,WAY 327157

5-HT3 antagonist 5 is a quinoxalin-2-carboxamide compound which is a 5-HT 3 receptor antagonist. 5-HT3 antagonist 5 exerts antagonism on 5-HT 3 agonist and 2-methyl-5-HT, and exhibits anti-depressant effect in mice [1].

价 格：￥电议型 号：T9846产 地：中国大陆

T9786Lu AF27139Inhibitor,P2XRs,oral,P2X7,rodent-active,Lu AF 27139,CNS-penetrant,CNS,Lu AF27139,Lu AF-271

Lu AF27139 is an effective and selective antagonist of P2X7 receptor (IC50s of 12 and 2.4 nM for human and rat, Kis of 22, 54, and 13 nM for mouse, human, and rat, respectively). Lu AF27139 can be used in CNS diseases studies.

价 格：￥电议型 号：T9786产 地：中国大陆

TMO27134(3H)-QuinazolinoneInhibitor,Bacterial,4(3H)-Quinazolinone,4(3H)Quinazolinone,inhibit,4(3H) Quinazol

Some 4-quinazolinone derivatives have antiplatelet activity.

价 格：￥电议型 号：TMO2713产 地：中国大陆

T7130Navarixininhibit,CXC chemokine receptors,Inhibitor,MK 7123,Navarixin,SCH527123,SCH-527123,MK7123,CXC

Navarixin(SCH527123) is a novel, selective CXC chemokine receptor 2(CXCR2) antagonist that inhibits neutrophil activation and modulates neutrophil trafficking in animal models, characteristics that may be beneficial in the treatment of conditions with unbalanced pulmonary neutrophilia.

价 格：￥电议型 号：T7130产 地：中国大陆

T4118SB 271046 hydrochlorideoral,test,Serotonin Receptor,SB271046,5-HT Receptor,Inhibitor,inhibit,5-hydro

SB 271046 hydrochloride is selective, orally active 5-HT6 antagonist (pKi values are 9.02-8.92, 6.35, 6.55, 6.27 at 5-HT6, 5-HT1A, 5-HT1D and D3, and 6.05, 5.95, 5.76, 5.73, 5.62, 5.55, 5.41, 5.39, 5.27 and < 4.99 at 5-HT1B, 5-HT1F, α1B, 5-HT2C, 5-HT2A, D2, 5-HT2B, 5-HT7, 5-HT4 and 5-HT1E respectively) and is > 200-fold selective over 55 other receptors, enzymes and ion channels. It increases extracellular aspartate and glutamate in the frontal cortex and exhibits anticonvulsant activity (EC50:

价 格：￥电议型 号：T4118产 地：中国大陆

T7005UlixertinibERK,VRT 752271,Ulixertinib,inhibit,VRT-752271,BVD 523,BVD523,Inhibitor,Extracellular sign

Ulixertinib (BVD-523, VRT752271) is an effective and reversible ERK1/ERK2 inhibitor. The IC50 of Ulixertinib is less than 0.3 nM for ERK2.

价 格：￥电议型 号：T7005产 地：中国大陆

T14271Aminooxy-PEG4-alcoholAminooxy PEG4 alcohol,AminooxyPEG4alcohol,Aminooxy-PEG-4-alcohol

Aminooxy-PEG4-alcohol is both a non-cleavable 4-unit PEG ADC linker and a PEG-based PROTAC linker.

价 格：￥电议型 号：T14271产 地：中国大陆

T10381AS2717638AS2717638,AS-2717638

AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5). It also significantly improves PGF2α-, PGE2-, and AMPA-induced allodynia.

价 格：￥电议型 号：T10381产 地：中国大陆

TP1925LtcY-NH2 TFA(327177-34-4 free base)tcY-NH-2 TFA(327177-34-4 free base),tcY NH2 TFA(327177 34 4 free b

tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.

价 格：￥电议型 号：TP1925L产 地：中国大陆

T6271TipifarnibZarnestra；IND 58359；R115777；替吡法尼

Tipifarnib is a nonpeptidomimetic quinolinone with potential antineoplastic activity. Tipifarnib binds to and inhibits the enzyme farnesyl protein transferase, an enzyme involved in protein processing (farnesylation) for signal transduction. By inhibiting

价 格：￥电议型 号：T6271产 地：中国大陆