T16536Pimonidazole hydrochlorideinhibit,Pimonidazole hydrochloride,Pimonidazole,Inhibitor

Pimonidazole hydrochloride accumulates in hypoxic cells via covalent binding with macromolecules or by forming reductive metabolites after the reduction of its nitro group. It can be used for qualitative and quantitative assessment of tumor hypoxia. Pimonidazole hydrochloride is a novel hypoxia marker for the complementary study of tumor hypoxia and cell proliferation in tumors.

价 格：￥电议型 号：T16536产 地：中国大陆

T5373Acrizanib

Acrizanib is a VEGFR-2 inhibitor, with an IC50 of 17.4 nM for BaF3-VEGFR-2.

价 格：￥电议型 号：T5373产 地：中国大陆

T61518TAK-653

TAK-653, an AMPA receptor potentiator with minimal agonistic activity, produces an antidepressant-like effect with a favorable safety profile in rats.

价 格：￥电议型 号：T61518产 地：中国大陆

T6582Mezlocillin SodiumBAY-f 1353,Mezlocillin Sodium,bacterial infection,gram-positive bacteria,Mezlocill

Mezlocillin sodium is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positive, organisms.

价 格：￥电议型 号：T6582产 地：中国大陆

T9353OXOMEMAZINEhistamine H1-receptor,OXOMEMAZINE,Histamine Receptor,inhibit,phenothiazine,antimuscarinic

Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low (Ki=1.65 μM, M2 receptors) affinity sites 20 times the difference[1]. Oxomemazine is an antihistamine and anticholinergic agent used in studies related to cough studies[2].

价 格：￥电议型 号：T9353产 地：中国大陆

T7703PK11007PK11007,inhibit,MDM-2/p53,Reactive Oxygen Species,Inhibitor,PK 11007,PK-11007

PK11007 is an anti-p53 drug.

价 格：￥电议型 号：T7703产 地：中国大陆

TN1539Cussosaponin CCussosaponin C,Inhibitor,inhibit

Cussosaponin C is a natural product isolated from Pulsatilla koreana Nakai.

价 格：￥电议型 号：TN1539产 地：中国大陆

T6965RG7112E1 activating enzyme,Inhibitor,RO-5045337,E1/E2/E3 Enzyme,RG7112,Ubiquitin conjugating enzyme,

RG7112 (RO5045337) is an orally bioavailable and selective p53-MDM2 inhibitor.

价 格：￥电议型 号：T6965产 地：中国大陆

T23074NNC 63-0532

NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.

价 格：￥电议型 号：T23074产 地：中国大陆

Fr12535Compound Fr12535Compound Fr12535

价 格：￥电议型 号：Fr12535产 地：中国大陆

T25534Indazole-Cl

Indazole-Cl is a selective ER? agonist and a selective estrogen receptor modifier (SERM).

价 格：￥电议型 号：T25534产 地：中国大陆

T67742EX-A5386

EX-A5386 is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.

价 格：￥电议型 号：T67742产 地：中国大陆

TP1086Men 10376 TFA(135306-85-3,free)Men 10376 TFA(135306853,free),Men 10376 TFA(135306 85 3,free)

Men 10376 TFA is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.

价 格：￥电议型 号：TP1086产 地：中国大陆

Fr14534Compound Fr14534Compound Fr14534

价 格：￥电议型 号：Fr14534产 地：中国大陆

T9753LEI110HepG2 cells,inhibit,thiol hydrolases,LEI110,Inhibitor,LEI-110,lipolysis,Phospholipase,LEI 110

LEI110 is a potent Phospholipase A2, group XVI (PLA2G16) inhibitor with an Ki value of 20 nM. LEI110 is a selective pan-inhibitor of the HRASLS family of thiol hydrolases (i.e., PLA2G16, HRASLS2, RARRES3 and iNAT).

价 格：￥电议型 号：T9753产 地：中国大陆

T13353Xanomeline oxalate

Xanomeline oxalate is a potent and selective muscarinic receptor agonist (SMRA) and stimulates phosphoinositide hydrolysis in vivo. Xanomeline oxalate can be used for the research of Alzheimer’s disease.

价 格：￥电议型 号：T13353产 地：中国大陆

T15388GLPG0974

GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.

价 格：￥电议型 号：T15388产 地：中国大陆

T8592CTK8A3536CTK-8A3536,CTK8A3536

CTK8A3536 is an inhibitor of Androgen receptor.

价 格：￥电议型 号：T8592产 地：中国大陆

T5362Y06036inhibit,Epigenetic Reader Domain,Inhibitor,Y-06036,Y 06036,Y06036

Y06036, a potent and selective BET inhibitor, can bind to the BRD4(1) bromodomain (Kd: 82 nM).

价 格：￥电议型 号：T5362产 地：中国大陆

TMA05362-Acetylbenzoic acid2 Acetylbenzoic acid,2Acetylbenzoic acid

2-Acetylbenzoic acid is more potent than 2-propionyloxybenzoic acid in inhibiting platelet function and platelet prostaglandin (PG) synthesis although the potencies of these agents were comparable in inhibiting prostacyclin (PGI2) synthesis.

价 格：￥电议型 号：TMA0536产 地：中国大陆