当前位置:易推广 > 上海陶术生物科技有限公司 > 产品展示
企业档案
会员类型:会员
已获得易推广信誉 等级评定
(0 -40)基础信誉积累,可浏览访问
(41-90)良好信誉积累,可接洽商谈
(91+ )优质信誉积累,可持续信赖
易推广会员:5年
最后认证时间:
注册号: 【已认证】
法人代表: 【已认证】
企业类型:生产商 【已认证】
注册资金:人民币万 【已认证】
产品数:86101
参观次数:3547116
已选条件
-
T7361Verucerfont;化合物VerucerfontNBI77860|||GSK561679;NBI77860|||3-(4-甲氧基-2-甲基苯基)-2,5-二甲基-N-[(1S)-1-(3-甲基-1
Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .
价 格:¥电议型 号:T7361产 地:中国大陆
-
T7337Kinetin riboside动力精核苷N6-Furfuryladenosine|||动力精核苷
Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)
价 格:¥电议型 号:T7337产 地:中国大陆
-
T72827Nrf2/HO-1-IN-1;化合物 Nrf2/HO-1-IN-1Nrf2/HO-1-IN-1
Nrf2/HO-1-IN-1 is a potent Nrf2/HO-1 pathway inhibitor, with an IC 50 value of 0.38 μM for NO . Nrf2/HO-1-IN-1 can significantly reduce the level of ROS in cells. Nrf2/HO-1-IN-1 can be used for researching anti-inflammatory [1] .
价 格:¥电议型 号:T72827产 地:中国大陆
-
T72760Keap1-Nrf2-IN-6;化合物 Keap1-Nrf2-IN-6Keap1-Nrf2-IN-6
Keap1-Nrf2-IN-6 is a potent, selective inhibitor of the Keap1-Nrf2 protein?protein interaction (PPI), demonstrating an inhibitory concentration (IC50) of 41 nM and a dissociation constant (Kd) of 68 nM.
价 格:¥电议型 号:T72760产 地:中国大陆
-
T72706Keap1-Nrf2-IN-13;化合物 Keap1-Nrf2-IN-13Keap1-Nrf2-IN-13
Keap1-Nrf2-IN-13 is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), exhibiting an IC50 value of 0.15 μM, indicative of its high efficacy. It binds strongly to the Keap1 protein by forming hydrogen bonds with critical polar residues (Asn414, Arg415, Arg483, Gln530), showcasing its specificity. This compound has implications for research into diseases associated with oxidative stress and inflammation, such as pulmonary fibrosis, chronic obstructive pulmonary disorder (COPD)
价 格:¥电议型 号:T72706产 地:中国大陆
-
T72697Nrf2 activator-6;化合物 Nrf2 activator-6Nrf2 activator-6
Nrf2 Activator-6, a tetrahydroisoquinoline compound, functions as an Nrf2 activator, demonstrating potency with an IC50 value of 5 nM in inhibiting the Kelch domain-Nrf2 interaction.
价 格:¥电议型 号:T72697产 地:中国大陆
-
T72687Keap1-Nrf2-IN-11;化合物 Keap1-Nrf2-IN-11Keap1-Nrf2-IN-11
Keap1-Nrf2-IN-11 (Compound 6k), a potent Keap1-Nrf2 inhibitor, exhibits a dissociation constant (KD) of 0.21 nM. It hampers the production of reactive oxygen species (ROS) and nitric oxide (NO), as well as the expression of tumor necrosis factor-alpha (TNF-α). By promoting Nrf2 nuclear translocation, it mitigates inflammation and is utilized in anti-inflammatory studies [1].
价 格:¥电议型 号:T72687产 地:中国大陆
-
T72417AChE/Nrf2 modulator 1;化合物 AChE/Nrf2 modulator 1AChE/Nrf2 modulator 1
AChE/Nrf2 modulator 1, an orally active compound, serves as a modulator of acetylcholinesterase (AChE) and nuclear factor erythroid 2-related factor 2 (Nrf2). It exhibits Nrf2 inductive activity alongside inhibitory effects on eeAChE and hAChE, demonstrating IC 50 values of 0.07 μM and 0.38 μM, respectively. This compound is applicable in Alzheimer´s disease research.
价 格:¥电议型 号:T72417产 地:中国大陆
-
T71944FGF/PDGF/VEGF RTK Inhibitor;化合物 FGF/PDGF/VEGF RTK InhibitorFGF/PDGF/VEGF RTK Inhibitor
FGF/PDGF/VEGF RTK Inhibitor is a potent, reversible, atp-competitive inhibitor against pdgfrβ, fgfr-1, and vegfr-2 (ic50 = 20, 90, and 240 nm, respectively) and effectively suppresses vegf-stimulated proliferation of hmvecs (ec50 = 420 nm).
价 格:¥电议型 号:T71944产 地:中国大陆
-
T71821Norfenefrine HCl;化合物 Norfenefrine HClNorfenefrine HCl
Norfenefrine is an Adrenergic Agonist. It is used in the treatment of female stress incontinence.
价 格:¥电议型 号:T71821产 地:中国大陆
-
T71587Fluoxetine succinate ester;化合物 Fluoxetine succinate esterFluoxetine succinate ester
Fluoxetine succinate ester is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used for the treatment of major depressive disorder, obsessive–compulsive disorder, bulimia nervosa, panic disorder, and premenstrual dysphoric disorder.
价 格:¥电议型 号:T71587产 地:中国大陆
-
T71415FPL-63012AR;化合物 FPL-63012ARFPL-63012AR
FPL-63012AR is a D1-receptor agonist.
价 格:¥电议型 号:T71415产 地:中国大陆
-
T71302Norfluoxetine-d5 HCl;化合物 Norfluoxetine-d5 HClNorfluoxetine-d5 HCl
Norfluoxetine-d5 is intended for use as an internal standard for the quantification of norfluoxetine by GC- or LC-MS. Norfluoxetine is an active metabolite of the antidepressant fluoxetine. It is formed from fluoxetine by the cytochrome P450 (CYP) isoforms CYP2C9, CYP2C19, and CYP3A. Norfluoxetine inhibits serotonin (5-HT) uptake in rat brain synaptosomal membrane preparations (Ki = 44.7 nM) and isolated human platelets (IC50 = ~15 nM). It has been found in the tissues of fish exposed to wastewa
价 格:¥电议型 号:T71302产 地:中国大陆
-
T71177LCRF-0004;化合物 LCRF-0004LCRF-0004
LCRF-0004 is a potent and selective RON receptor tyrosine kinase inhibitor. The RON receptor tyrosine kinase has been identified as an important mediator of KRAS oncogene addiction and is overexpressed in the majority of pancreatic cancers. Preclinical studies show that inhibition of RON function decreases pancreatic cancer cell migration, invasion, and survival and can sensitize pancreatic cancer cells to chemotherapy. RON receptor tyrosine kinase is a potential as a therapeutic target.
价 格:¥电议型 号:T71177产 地:中国大陆
-
T71011Perfluorinated SAHA;化合物 Perfluorinated SAHAPerfluorinated SAHA
Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer.
价 格:¥电议型 号:T71011产 地:中国大陆
-
T70872Smurf1 inhibitor 1;化合物 Smurf1 inhibitor 1Smurf1 inhibitor 1
Smurf1 inhibitor 1 is a inhibitor that promotes bone formation.
价 格:¥电议型 号:T70872产 地:中国大陆
-
T70655Furaprevir;化合物 FuraprevirFuraprevir
Furaprevir is an HCV NS3/4A Inhibitor
价 格:¥电议型 号:T70655产 地:中国大陆
-
T70067IRFI-165;化合物 IRFI-165IRFI-165
IRFI-165 is an adenosine A1 receptor inhibitor
价 格:¥电议型 号:T70067产 地:中国大陆
-
T6S1500Ginsenoside Rf;人参皂苷 RfGinsenoside-Rf|||Panaxoside Rf;人参皂苷 Rf|||Ginsenoside-Rf|||Panaxoside Rf
Ginsenoside Rf (Panaxoside Rf) is a trace component of ginseng root. Ginsenoside Rf inhibits N-type Ca2+ channel.
价 格:¥电议型 号:T6S1500产 地:中国大陆
-
T69921BRF110;化合物 BRF110BRF110
BRF110 is a brain penetrant, potent and selective agonist of nuclear receptor-related 1 (Nurr1):Retinoid X receptor α (RXRα) heterodimer. BRF110 is a neuroprotective agent that prevents dopaminergic neuron demise and striatal dopaminergic denervation in vivo against PD-causing toxins. It induced dopamine biosynthesis in vivo. BRF110 chronic dosing does not induce dyskinesia in mice model.
价 格:¥电议型 号:T69921产 地:中国大陆