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T16688Pyr6；化合物Pyr6N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide；N-
Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx inhibition in thapsigargin depleted native RBL-2H3 cells).Pyr6 is an inhibitor of Ca2+ entry, which displays higher potency to inhibit Ca2+ entry mediated by CRAC channel than by TRPC3.
价 格：￥电议型 号：T16688产 地：中国大陆
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T16687Pyr3；化合物Pyr3Pyr3
Pyr3 is a selective transient receptor potential canonical channel 3 inhibitor. Pyr3 inhibits TRPC3-mediated Ca2+ influx in a dose-dependent manner(IC50 = 700 nM).
价 格：￥电议型 号：T16687产 地：中国大陆
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T16686Pyr10；化合物Pyr10Pyr10
Pyr10 is a pyrazole derivative and a selective TRP cation 3 inhibitor. Pyr10 has the ability to distinguish between receptor-operated TRPC3 and native stromal interaction molecule 1 (STIM1)/Orai1 channels. Pyr10 inhibits Ca2+ influx in carbachol-stimulated TRPC3-transfected HEK293 cells (IC50: 0.72 μM) (IC50 of 13.08 μM for store-operated Ca2+ entry in BRL-2H3 cells) .
价 格：￥电议型 号：T16686产 地：中国大陆
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T16685Purpurogallin红倍酚红倍酚|||红陪酚
Purpurogallin is a naturally phenol extracted from the plants of Quercus spp. It has effective xanthine oxidase inhibitory activity (IC50: 0.2 μM). Purpurogallin also has antioxidant and anti-inflammatory effects.
价 格：￥电议型 号：T16685产 地：中国大陆
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T16684Puromycin aminonucleoside维生素E醋酸酯维生素E醋酸酯|||NSC 3056
Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner.
价 格：￥电议型 号：T16684产 地：中国大陆
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T16683Pumosetrag Hydrochloride化合物 T16683MKC-733|||DDP-733
Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.
价 格：￥电议型 号：T16683产 地：中国大陆
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T16682Pumaprazole；普马拉唑BY-841；BY-841|||普马拉唑
Pumaprazole (BY-841) is an antagonist of a reversible proton pump.
价 格：￥电议型 号：T16682产 地：中国大陆
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T16681Nesolicaftor；化合物PTI-428PTI-428；PTI-428
Nesolicaftor (PTI-428) specifically enhances cystic fibrosis transmembrane conductance regulator protein synthesis.
价 格：￥电议型 号：T16681产 地：中国大陆
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T16680PTC-028；化合物PTC-028PTC-028
PTC-028 selectively suppresses cancer cells whereas normal cells remain unaffected. PTC-028 is an orally bioavailable inhibitor of stem cell factor BMI-1 in ovarian cancer. The depletion of BMI-1 by PTC-028 causes caspase-mediated apoptosis.
价 格：￥电议型 号：T16680产 地：中国大陆
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T1668Vinblastine sulfate；硫酸长春碱NSC49842|||Vincaleukoblastine sulfate salt；硫酸长春碱|||NSC49842|||Vincaleukobla
Vinblastine sulfate (Vincaleukoblastine sulfate salt) can inhibit the formation of microtubule, it also inhibits nAChR(IC50=8.9 uM).
价 格：￥电议型 号：T1668产 地：中国大陆
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T16679Belzutifan；化合物BelzutifanPT2977|||MK-6482；PT2977|||MK-6482
Belzutifan (MK-6482) is a potential treatment for clear cell renal cell carcinoma (ccRCC). Belzutifan is an orally active and selective HIF-2α inhibitor (IC50: 9 nM). Belzutifan , as a second-generation HIF-2α inhibitor, increases potency and improves pharmacokinetic profile.
价 格：￥电议型 号：T16679产 地：中国大陆
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T16678PSN632408；化合物 T16678PSN632408
PSN632408 is an optimized agonist of GPR119 receptors that display similar potency to OEA at both recombinant mouse and human GPR119 receptors (EC50: 5.6 and 7.9 uM, respectively).
价 格：￥电议型 号：T16678产 地：中国大陆
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T16677Psicofuranine；化合物 T16677Psicofuranine
Psicofuranine also specifically inhibits GMP synthase and interrupts parasite growth. Psicofuramine is a nucleoside antibiotic. It has the inhibition of xanthosine 5´-phosphate aminase. Psicofuranine shows dose-dependent inhibition of P. falciparum growth(IC50: 0.3 mM).
价 格：￥电议型 号：T16677产 地：中国大陆
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T16676PSI-697；化合物 T16676P-Selectin Inhibitor；P-Selectin Inhibitor
PSI-697 is an inhibitor of oral P-selectin (IC50: 125 μM).
价 格：￥电议型 号：T16676产 地：中国大陆
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T16674Pseudouridine；假尿苷Pseudouridine
Pseudouridine is the most abundant modified nucleoside in non-coding RNAs. It enhances the function of transfer RNA and ribosomal RNA by stabilizing RNA structure.
价 格：￥电议型 号：T16674产 地：中国大陆
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T16673Pseudouridimycin；化合物 T16673PUM；PUM
Pseudouridimycin is a C-nucleoside analogue. Pseudouridimycin is an antibiotic and is a selective bacterial RNA polymerase (RNAP) inhibitor. It is effective against both Gram-negative and Gram-positive bacteria.
价 格：￥电议型 号：T16673产 地：中国大陆
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T16672PSB-1114 tetrasodium；化合物 T16672PSB-1114 tetrasodium
PSB-1114 tetrasodium shows >50-fold selectivity versus the P2Y4 (EC50: 9.3 μM) and P2Y6 (EC50: 7.0 μM) receptors. PSB-1114 tetrasodium is an effective, enzymatically stable, and subtype-selective P2Y2 receptor agonist (EC50: 134 nM) .
价 格：￥电议型 号：T16672产 地：中国大陆
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T16671PS315；化合物 T16671PS315
PS315 inhibits the full-length and catalytic domain constructs of PKCζ (IC50=10 μM) and PKCη (IC50=30 μM). PS315 has anti-cancer activity. PS315 is a derivative of PS48 and is an allosteric PKC inhibitor by binding to the PIF-pocket of aPKC and inducing displacement of the active site residue Lys111.
价 格：￥电议型 号：T16671产 地：中国大陆
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T16670PS210；化合物PS210PS210
PS210 is a potent and selective activator of PDK1 (Kd: 3 μM), specifically targeting the PIF-binding pocket of PDK1, without acting against other protein kinases such as S6K, PKB/Akt, or GSK3. Its prodrug, PS423, serves as a substrate-selective inhibitor of PDK1 in cells, inhibiting the phosphorylation and activation of S6K.
价 格：￥电议型 号：T16670产 地：中国大陆
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T1667Tandutinib；坦度替尼MLN518|||CT53518|||NSC726292；MLN518|||CT53518|||NSC726292|||坦度替尼
Tandutinib (CT53518) (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit and PDGFR, 15-20 fold higher potency for FLT3 versus CSF-1R and >100-fold selectivity for the same target versus FGFR, EGFR, and KDR.
价 格：￥电议型 号：T1667产 地：中国大陆
