T9707DB2313

DB2313 is a potent transcription factor PU.1 inhibitor, IC50=14 nM. DB2313 disrupts the interaction of PU.1 with target gene promoters. DB2313 induces apoptosis of acute myeloid leukemia (AML) cells, and has anticancer effects

价 格：￥电议型 号：T9707产 地：中国大陆

T7549Talnetantschizophrenia,SB223412,NK receptor,Inhibitor,hNK-2,Talnetant,Neurokinin Receptor,Tachykinin

Talnetant is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission

价 格：￥电议型 号：T7549产 地：中国大陆

T6571Lomerizine dihydrochlorideCa2+ channels,Ca channels,inhibit,Lomerizine,KB 2796,KB2796,Lomerizine dih

Lomerizine dihydrochloride is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.

价 格：￥电议型 号：T6571产 地：中国大陆

T6S1367Procyanidin B2inhibit,Procyanidin B2,Proanthocyanidin B 2,Procyanidin B 2,Inhibitor,Proanthocyanidin

Procyanidin B2 has vascular protective, anti-diabetic nephropathy, anti-cancer, anti-inflammatory, and antioxidant activities. Procyanidin B2 inhibited NLRP3 inflammasome activation via suppression of AP-1 pathway.

价 格：￥电议型 号：T6S1367产 地：中国大陆

T6976SB 239063inhibit,SB 239063,SB-239063,Inhibitor,Autophagy,p38 MAPK

SB239063 is a potent and selective p38 MAPKα/β inhibitor with IC50 of 44 nM, showing no activity against the γ- and δ-kinase isoforms.

价 格：￥电议型 号：T6976产 地：中国大陆

T9230KM 91104V-ATPase human HSC,a3-b2 subunits,KM-91104,KM 91104,Inhibitor,KM91104,Proton Pump,cell-perme

KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.

价 格：￥电议型 号：T9230产 地：中国大陆

T10445B220B-220,B220

B220, an antiviral agent, inhibits the growth of HSV-1, HSV-2, and human cytomegalovirus (CMV).

价 格：￥电议型 号：T10445产 地：中国大陆

TJS0502Ilexsaponin B2Ilexsaponin B2

价 格：￥电议型 号：TJS0502产 地：中国大陆

T9687MAGL-IN-4Monoacylglycerol lipase,CB1,lipase,monoacylglycerol,CB2,Inhibitor,inhibit,BBB,barrier,MAGLI

MAGL-IN-4 is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.

价 格：￥电议型 号：T9687产 地：中国大陆

T7678SJB2-043SJB2-043,inhibit,DUBs,SJB2043,SJB-2-043,SJB2 043,Deubiquitinase,Inhibitor

SJB2-043 is an inhibitor of USP1-UAF1 ( IC50 : 544 nM).

价 格：￥电议型 号：T7678产 地：中国大陆

T6638RetapamulinRetapamulin,Bacterial,SB 275833,inhibit,SB275833,Inhibitor,Antibiotic

Retapamulin, a Pleuromutilin Antibacterial, binds to both E. coli and S. aureus ribosomes with similar potencies (Kd: 3 nM).

价 格：￥电议型 号：T6638产 地：中国大陆

T6713Ulipristalemergency,Deacetyl CDB2914,inhibit,contraception,CDB 3236,Progesterone Receptor,CDB3236,De

Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.

价 格：￥电议型 号：T6713产 地：中国大陆

T8839ICCB280ICCB 280,Inhibitor,ICCB280,Apoptosis,differentiation,proliferation,C/EBPα,anti-leukemic,ICCB-

ICCB280 was capable of inducing differentiation and apoptosis of ATRA-resistant patient blasts strongly signify that the activity of this compound can overcome resistance to other current therapies for AML with an unfavorable prognosis.

价 格：￥电议型 号：T8839产 地：中国大陆

T67747CB2R/FAAH modulator-3CB2R/FAAHmodulator3

CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 has research value related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.

价 格：￥电议型 号：T67747产 地：中国大陆

T7138FB23-2FB23 2,AML,Apoptosis,leukemia,acute,anti-proliferation,Inhibitor,FB232,m6A,myeloid,mRNA,inhibi

FB23-2 is a potent and selective mRNA N6-methyladenosine (m6A) demethylase FTO inhibitor(IC50 : 2.6 μM).

价 格：￥电议型 号：T7138产 地：中国大陆

T9194UMB298UMB-298,UMB298,inhibit,MOLM13,Inhibitor,bromodomain,UMB 298,selective,potent,Epigenetic Reader

UMB298 is a potent and selective CBP/P300 bromodomain inhibitor. UMB298 inhibits BRD4 with IC50 of 5193nM.

价 格：￥电议型 号：T9194产 地：中国大陆

T4671BN82002CDC25C,BN82002,CDC25A,BN-82002,inhibit,CDC25B3,MIA PaCa-2,Inhibitor,CDC25B2,BN 82002,Phosphat

BN82002 is a synthetic inhibitor of CDC25 phophatases

价 格：￥电议型 号：T4671产 地：中国大陆

T8874FB23Inhibitor,FB 23,FB-23,inhibit,anti-proliferative,demethylase,leukemogenesis,FTO,N6-methyladenosi

FB23 directly binds to FTO and selectively inhibits FTO´s m6A demethylase activity. (FTO, an mRNA N6-methyladenosine (m6A) demethylase, was reported to promote leukemogenesis.)

价 格：￥电议型 号：T8874产 地：中国大陆

T7671Myosminea4b2,Inhibitor,Myosmine,alkaloid,acetylcholinergic,nicotinic,receptors,Nicotinic acetylcholi

Myosmine is a minor tobacco alkaloid that is structurally related to nicotine.

价 格：￥电议型 号：T7671产 地：中国大陆

T10696CB2 modulator 1CB2 modulator 1,ischemia,CB-2 modulator 1,osteoporosis,CB2,inflammation,immunedisorde

CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.

价 格：￥电议型 号：T10696产 地：中国大陆