T8927WWL 154FAAH-4,Fatty acid amide hydrolase,Inhibitor,inhibit,WWL154,JZL184,WWL 154,FAAH

WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.

价 格：￥电议型 号：T8927产 地：中国大陆

T9611PF-04802367PF367,PF 367,protein,disease,Alzheimer,PF-04802367,PF-367,Glycogen synthase kinase-3,kina

PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay. It shows desirable central nervous system (CNS) properties and potency. It is equally effective at inhibition of the two known GSK-3 isoforms (GSK-3α and GSK-3β) with IC50 values of 10.0 and 9.0 nM in mobility shift assays, respectively.

价 格：￥电议型 号：T9611产 地：中国大陆

TN2030P-Hydroxyphenethyl trans-ferulateGlucosidase,inhibit,P Hydroxyphenethyl trans ferulate,Inhibitor,PHy

P-Hydroxyphenethyl trans-ferulate exhibits affinity toward 5-HT(7) receptors in a competitive binding assay. P-Hydroxyphenethyl trans-ferulate can double quinone reductase specific activity in Hepa 1c1c7 cells at a level of 2.1 microg/mL (6.6 microM).

价 格：￥电议型 号：TN2030产 地：中国大陆

T6956LProtirelin Acetate(24305-27-9 free base)Protirelin Acetate(24305279 free base),Protirelin Acetate(24

Protirelin Acetate is a tripeptide that stimulates the release of thyrotropin and prolactin.

价 格：￥电议型 号：T6956L产 地：中国大陆

T7149S29434cell-permeable,inhibit,selective,S 29434,HepG2,mice,NMDPEF,S-29434,ROS,Autophagy,S29434,Inhibi

S29434 (NMDPEF) is a potent, competitiveinhibitor of quinone reductase 2 (QR2;IC50:5-16nM).

价 格：￥电议型 号：T7149产 地：中国大陆

T6938PF-4989216Apoptosis,inhibit,Phosphoinositide 3-kinase,PF4989216,PF-4989216,PI3K,Inhibitor

PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.

价 格：￥电议型 号：T6938产 地：中国大陆

T6948Pluripotininhibit,Extracellular signal regulated kinases,Ribosomal S6 Kinase (RSK),SC-1,SC 1,Inhibit

Pluripotin (SC1), which keep embryonic stem cell (ESC) self-renewal, is a dual inhibitor of extracellular signal-regulated kinase 1 (ERK1, MAPK3) and RasGAP.

价 格：￥电议型 号：T6948产 地：中国大陆

T6409ALK kinase inhibitor-1kinase,ALK tyrosine kinase receptor,Anaplastic lymphoma kinase,lymphoma,Anapla

价 格：￥电议型 号：T6409产 地：中国大陆

TQ0055AMG-3969Hexokinase IV,AMG 3969,Hexokinase D,Glucokinase,Inhibitor,AMG3969,AMG-3969,inhibit

AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).

价 格：￥电议型 号：TQ0055产 地：中国大陆

TQ0232UNC0646H3K9me2,KMT1D,chromatin,EHMT1,Histone Methyltransferase,UNC-0646,SAR,inhibit,G9a,GLP,PKMT,UNC

UNC 0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50s: 6 nM/15 nM for G9a/GLP). UNC0646 potently blocks G9a/GLP methyltransferase activity in cells (IC50: 10 nM in MCF7 cells); exhibits low cellular toxicity (EC50: 4.7 μM in MCF7 cells).

价 格：￥电议型 号：TQ0232产 地：中国大陆

TN1134Euscaphic acidEuscaphic acid,Inhibitor,PI3K,inhibit,Apoptosis,Phosphoinositide 3-kinase,DNA/RNA Synt

Euscaphic acid has anti-diabetic, and anti-inflammatory activities, it inhibits LPS-induced inflammatory responses by interference with the clustering of TRAF6 with IRAK1 and TAK1, resulting in blocking the activation of IKK and MAPKs signal transduction to downregulate NF-κB activations.

价 格：￥电议型 号：TN1134产 地：中国大陆

T7041DonepezilE 2020,AChE,Donepezil,Cholinesterase (ChE),Inhibitor,E-2020,inhibit,hAChE,bAChE

Donepezil is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE). It can be used for the treatment of mild to moderate dementia of the Alzheimer´s type.

价 格：￥电议型 号：T7041产 地：中国大陆

T9003CVT-11127Inhibitor,apoposis,GS 456332,S-phase,monounsaturated fatty acids (MUFA),Stearoyl-CoA Desatu

CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.

价 格：￥电议型 号：T9003产 地：中国大陆

TN1405Arnicolide DMammalian target of Rapamycin,Phosphoinositide 3-kinase,inhibit,Inhibitor,Caspase,mTOR,A

Arnicolide D is a sesquiterpene lactone. Arnicolide D isolates from Centipeda minima. Arnicolide D modulates the cell cycle, activates the caspase signaling pathway and inhibits the PI3K/AKT/mTOR and STAT3 signaling pathways. Arnicolide D inhibits Nasopharyngeal carcinoma (NPC) cell viability in a concentration- and time-dependent manner. Arnicolide D exerts strong cytotoxic activity on the human colon carcinoma HT-29 cell line.

价 格：￥电议型 号：TN1405产 地：中国大陆

TP1772LHemokinin 1 (mouse) acetate(208041-90-1 free base)Hemokinin 1 (mouse) acetate(208041901 free base),H

Hemokinin 1 (mouse) acetate is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.

价 格：￥电议型 号：TP1772L产 地：中国大陆

T6S1485Ginsenoside Rh4Ginsenoside Rh-4,Ginsenoside Rh4

1. Ginsenoside Rh4 could be safely used as adjuvant with low or non-haemolytic effect. 2. Ginsenoside Rh4 has cytotoxic activity and its aglycone against cancer cell lines.

价 格：￥电议型 号：T6S1485产 地：中国大陆

T6S1500Ginsenoside RfCa channels,Calcium Channel,Ginsenoside Rf,Ca2+ channels,Endogenous Metabolite,Inhibit

Ginsenoside Rf is a trace component of ginseng root. Ginsenoside Rf inhibits N-type Ca2+ channel.

价 格：￥电议型 号：T6S1500产 地：中国大陆

TP1796Albiglutide TFA (782500-75-8 free base)Albiglutide TFA (782500758 free base),Albiglutide TFA (782500

Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).

价 格：￥电议型 号：TP1796产 地：中国大陆

T9215ELOVL6-IN-2ELOVL6IN2,ELOVL6 IN 2,plasma,inhibit,selective,ELOVL-6-IN-2,liver,dose-proportionally,Inh

ELOVL6-IN-2 is a orally active and selective ELOVL6 inhibitor.

价 格：￥电议型 号：T9215产 地：中国大陆

TP1992LM40 acetate(143896-17-7 free base)M-40 acetate(143896-17-7 free base),M40 acetate(143896 17 7 free b

M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat brain in vitro (IC50 = 3 - 15 nM). Attenuates the antidepressant effects of fluoxetine and blocks galanin-induced food intake in vivo. Also exhibits weak partial agonist activity at peripheral GAL2 receptors at doses > 100 nM.

价 格：￥电议型 号：TP1992L产 地：中国大陆