T6727VU0364770inhibit,Metabotropic glutamate receptors,VU0364770,VU-0364770,Inhibitor,mGluR

VU 0364770(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu subtypes.

价 格：￥电议型 号：T6727产 地：中国大陆

T67709HispolonHISPOLON(P)

Hispolon is a polyphenol. Hispolon can be isolated from Phellinus linteus. Hispolon exhibits anticancer, antidiabetic, antiviral, hepatoprotective, antioxidant, and anti-inflammatory activities.

价 格：￥电议型 号：T67709产 地：中国大陆

T6126JNJ-7706621JNJ7706621；JNJ 7706621

JNJ-7706621 is a potent aurora kinase inhibitor, and also inhibits CDK1 and CDK2.

价 格：￥电议型 号：T6126产 地：中国大陆

T6027Delanzomib德兰佐米；CEP-18770

CEP-18770 is an orally active inhibitor of the chymotrypsin-like activity of proteasome (IC50: 3.8 nM). It only marginally inhibits the tryptic and peptidylglutamyl activities of the proteosome.

价 格：￥电议型 号：T6027产 地：中国大陆

T5770Alisol B

Alisol B may be a potential novel therapeutic molecule for bone disorders through targeting the differentiation of osteoclasts as well as their functions. Alisol B also inhibited RANKL-induced expression of NFATc1 and c-Fos, which are key transcription fa

价 格：￥电议型 号：T5770产 地：中国大陆

T47703-Amino-4-hydroxybenzoic acid3-氨基-4-羟基苯甲酸；3-amino-4-hydroxybenzenecarboxylic acid

3-Amino-4-hydroxybenzoic acid is a useful research chemical.

价 格：￥电议型 号：T4770产 地：中国大陆

T377092,2,2-Trichloroethanol

2,2,2-Trichloroethanol is an agonist of the nonclassical K2P channels TREK-1 and TRAAK.

价 格：￥电议型 号：T37709产 地：中国大陆

T3770Taraxasterol蒲公英甾醇；Taraxasterin

Taraxasterol is compound with anti-inflammatory activity.

价 格：￥电议型 号：T3770产 地：中国大陆

T2O2770Agarotetrol

价 格：￥电议型 号：T2O2770产 地：中国大陆

T2996TetrandrineNSC-77037；d-Tetrandrine；Sinomenine A；Fanchinine；Hanfangchin A；粉防己碱；汉防己甲素

Tetrandrine is a natural, bis-benzylisoquinoline alkaloid isolated from the root of the plant. Tetrandrine non-selectively inhibits calcium channel activity and induces G1 blockade of the G1 phase of the cell cycle and apoptosis in various cell types, res

价 格：￥电议型 号：T2996产 地：中国大陆

T2770Gentiopicroside龙胆苦甙；龙胆苦苷；Gentiopicrin

Gentiopicroside, a naturally occurring iridoid glycoside, extracted from Gentiana manshurica Kitag, inhibits P450 activity, with an IC50 and a Ki of 61 μM and 22.8 μM for CYP2A6; has antianti-inflammatoryand antioxidative effects.

价 格：￥电议型 号：T2770产 地：中国大陆

T2588IvacaftorIvacaftor (VX-770)；VX-770；依伐卡托

Ivacaftor (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells, respectively.

价 格：￥电议型 号：T2588产 地：中国大陆

T2386Pirfenidone吡非尼酮；S-7701,AMR-69；AMR69；S-7701

Pirfenidone is an inhibitor for TGF-β production and TGF-β stimulated collagen production. Pirfenidone inhibits fibroblast, epidermal, platelet-derived, and transforming beta-1 growth factors, thereby slowing tumor cell proliferation. This agent also inhi

价 格：￥电议型 号：T2386产 地：中国大陆

T21059Ticagrelor metabolite M5替格瑞洛杂质H；Ticagrelor metabolite M5,；T437700；AR-C133913XX

Ticagrelor metabolite M5 is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor. Compared to Clopidogrel, Ticagrelor has faster and more consistent inhibition on ADP-receptors. Ticagrelor is used in the treatment of acute co

价 格：￥电议型 号：T21059产 地：中国大陆

T20770BAY32-59158-羟基喹啉-2-羧酸；BAY 32 5915；BAY 32-5915；BAY32 5915；BAY-32-5915；BAY325915

BAY32-5915 is a selective inhibitor of IKKalpha.

价 格：￥电议型 号：T20770产 地：中国大陆

T1923BRD4770

BRD4770 is a histone methyltransferase G9a inhibitor and induces cell senescence.

价 格：￥电议型 号：T1923产 地：中国大陆

T1770GNE-9605GNE9605

GNE-9605 is a highly effective, specifical, and brain-penetrant LRRK2 inhibitor (IC50: 19 nM).

价 格：￥电议型 号：T1770产 地：中国大陆

T13017STL127705Compound L；7-[[2-(3,4-Dimethoxyphenyl)ethyl]amino]-3-(3-fluorophenyl)pyrimido[4,5-d]pyrimid

STL127705 is a potent Ku 70/80 heterodimer protein inhibitor and inhibits Ku70/80-DNA interaction with IC50 of 3.5 μM. STL127705 inhibits the activation of Ku-dependent DNA-PKCS kinase with IC50 of 2.5 μM.

价 格：￥电议型 号：T13017产 地：中国大陆

T1193Clomiphene citrate枸橼酸氯米芬；NSC 35770；Clomifene citrate

Clomifene Citrate is a selective estrogen receptor modulator.

价 格：￥电议型 号：T1193产 地：中国大陆

T11766LEltanexorKPT-8602；ONO-7706；ATG-016

Eltanexor is an orally active exportin-1 (XPO1) inhibitor. It has effective anti-leukemic activity. Eltanexor inhibits XPO1-dependent nuclear export (EC50=60.9 nM) by directly targeting XPO1. Eltanexor causes caspase-dependent apoptosis in a panel of leuk

价 格：￥电议型 号：T11766L产 地：中国大陆