T13314VTX-27Inhibitor,VTX27,VTX 27,PKC,Protein kinase C,inhibit,VTX-27

VTX-27 is a selective inhibitor of protein kinase C θ (PKC θ) (Kis: 0.08 nM and 16 nM for PKC θ and PKC δ).

价 格：￥电议型 号：T13314产 地：中国大陆

TQ0091LY2795050LY2795050,Inhibitor,central nervous system dysfunction,sex differences,inhibit,Opioid Recep

LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).

价 格：￥电议型 号：TQ0091产 地：中国大陆

T12784RWJ 63556

RWJ 63556 is an orally active inhibitor of COX-2 selective/5-lipoxygenase, shows anti-inflammatory activities.

价 格：￥电议型 号：T12784产 地：中国大陆

T8272TrierucinEndogenous Metabolite,Inhibitor,inhibit,Trierucin

Trierucin is a trierucic acid triglyceride isolated from the seed oil.

价 格：￥电议型 号：T8272产 地：中国大陆

T9272Xaliproden hydrochloride5-HT Receptor,Xaliproden hydrochloride,SR57746A,Serotonin Receptor,dopamine,

Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.

价 格：￥电议型 号：T9272产 地：中国大陆

TN12744-Allylcatechol4Allylcatechol,4-Allylcatechol,Inhibitor,inhibit,4 Allylcatechol

4-Allylpyrocatechol has antioxidant activity, it has protective activity against the photosensitization-induced damage to lipids and proteins of rat liver mitochondria, which attributes to its free radical and singlet oxygen scavenging properties.

价 格：￥电议型 号：TN1274产 地：中国大陆

T67727MCT1-IN-3MCT1IN3

MCT1-IN-3 is a monocarboxylate transporter 1 (MCT1) inhibitor. The solute carrier (SLC) monocarboxylate transporter 1 (MCT1; SLC16A1) represents a promising target for the treatment of cancer. MCT1-IN-3 (compound 24) showed the highest MCT1 transport inhibition with an IC50 value of 81.0 Nm. MCT1-IN-3 has also significant inhibitivity against the multidrug transporter ABCB1.

价 格：￥电议型 号：T67727产 地：中国大陆

TP1936L1RFRP3(human) acetate(311309-27-0 free base)RFRP-3(human) acetate(311309-27-0 free base),RFRP3(human)

RFRP-3(human) acetate, a human GnIH peptide homolog, is a potent inhibitor of gonadotropin secretion by inhibiting Ca2+ mobilization. RFRP-3(human) acetate is a NPFF1 receptor agonist, it inhibits forskolin-induced production of cAMP with an IC50 of 0.7 nM.

价 格：￥电议型 号：TP1936L1产 地：中国大陆

T8279Isobornyl acetateInhibitor,Isobornyl,Isobornyl acetate,inhibit

价 格：￥电议型 号：T8279产 地：中国大陆

TP1273FLAG peptideInhibitor,FLAG peptide,inhibit

FLAG peptide is an eight amino acids peptide (Asp-Tyr-Lys-Asp-Asp-Asp-Asp-Lys) with an enterokinase-cleavage site used for the purification of recombinant proteins.

价 格：￥电议型 号：TP1273产 地：中国大陆

TP1293Jagged-1 (188-204) TFA(219127-21-6 free base)Jagged1 (188204) TFA(219127216 free base),Jagged 1 (188

Jagged-1 (188-204) TFA is a fragment of the JAG-1 protein. JAG-1 is Notch ligand, a peptide that is the most conspicuously expressed ligand in skin. JAG-1 induces epidermal maturation. Exposing submerged keratinocytes monolayers to JAG-1 with elevated calcium concentration produces stratification with loricrin expression and NF-alphaB activation.

价 格：￥电议型 号：TP1293产 地：中国大陆

T16766Ro 08-2750growth,MSI,Ro 082750,p75NTR,TRKA,RNA-binding,Nerve,NGF,Inhibitor,leukemia,Apoptosis,AML,Ro

Ro 08-2750 is a non-peptide and reversible nerve growth factor (NGF) inhibitor which binds to NGF, and with an IC50 of ~ 1 ?M. Ro 08-2750 is a selective MSI RNA-binding activity inhibitor, with an IC50 of 2.7 μM. Ro 08-2750 inhibits NGF binding to p75NTR selectively over TRKA.

价 格：￥电议型 号：T16766产 地：中国大陆

T6837FlavopiridolHMR1275,inhibit,L86-8275,CDK,Cyclin dependent kinase,Inhibitor,Autophagy,HMR 1275,Human

Flavopiridol (Alvocidib) competes with ATP to inhibit CDKs including CDK1, CDK2, CDK4 and CDK6 with IC50 of ~ 40 nM. It is 7.5-fold more selective for CDK1, 2, 4, 6 versus CDK7. Flavopiridol is initially found to inhibit EGFR and PKA. Phase 1/2.

价 格：￥电议型 号：T6837产 地：中国大陆

T27093CT-1

CT-1 is a DNA minor groove ligand and causes p53-dependent breast cancer cell apoptosis.

价 格：￥电议型 号：T27093产 地：中国大陆

T9274antifungal-agent-6Inhibitor,Fungal,Antifungal agent6,inhibit,antifungalagent6,antifungal agent 6,Ant

Antifungal agent 6 shows antifungal activity.

价 格：￥电议型 号：T9274产 地：中国大陆

T6411BiapenemL627,inhibit,L-627,CLI86815,LJC10627,Bacterial,LJC-10627,Antibiotic,CLI-86815,Biapenem,Inhib

Biapenem is a 1-beta-methylcarbapenem antibiotic with a wide range of antibacterial activity. Biapenem has similar antibacterial activity to that of imipenem, but is more stable against human renal dehydropeptidase-I and with less neurotoxicity.

价 格：￥电议型 号：T6411产 地：中国大陆

TQ0027Transcrocetinate disodiumiGluR,Transcrocetinate disodium,Inhibitor,inhibit,Ionotropic glutamate rece

Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), is a high-affinity antagonist of NMDA receptor.

价 格：￥电议型 号：TQ0027产 地：中国大陆

T12753RORγt Inverse agonist 6Inhibitor,ROR,RORγt Inverse agonist-6,inhibit,RAR-related orphan receptor,ROR

RORγt Inverse agonist 6 is an agonist of RORγt inverse. RORγt Inverse agonist 6 can be used in research on Th17-driven autoimmune diseases.

价 格：￥电议型 号：T12753产 地：中国大陆

T64327Fmoc-Cys(Acm)-OH

Fmoc-Cys(Acm)-OH is a cysteine derivative.

价 格：￥电议型 号：T64327产 地：中国大陆

TQ0277PralsetinibInhibitor,BLU 667,BLU-667,Pralsetinib,inhibit,RET

Pralsetinib (BLU-667) is a highly potent, selective RET inhibitor (IC50s: 0.4, 0.3, 0.4, 0.4, and 0.4 nM for WT RET, RET mutants V804L, V804M, M918T and CCDC6-RET fusion).

价 格：￥电议型 号：TQ0277产 地：中国大陆