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(41-90)ۣɽǢ̸
(91+ )ۣɳ
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עţ ֤
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עʽ ֤
Ʒ86101
ι۴3752652
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Fr14055Compound Fr14055Compound Fr14055
ţFr14055 أй½
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T13246UCT943UCT-943,UCT943
UCT943 is an inhibitor of Plasmodium falciparum PI4K (IC50 = 23 nM).
ţT13246 أй½
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T75283,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate3,7dimethylocta2,6dienyl 5,9,13tr
3,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate is a chemical compound
ţT7528 أй½
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T6443Chloroprocaine hydrochlorideinhibit,Na,K-ATPase,Sodium potassium pump,Chloroprocaine,anesthetic,2-Ch
Chloroprocaine HCl is a local anesthetic during surgical procedures.
ţT6443 أй½
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T7596FirocoxibLPS,COX-2,fever,ML1785713,Cyclooxygenase,COX,inhibit,Firocoxib,Inhibitor,anti-inflammatory,
Firocoxib is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 M), with anti-inflammatory for use in dogs and horses.
ţT7596 أй½
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T60057WAY-388657WAY 388657,WAY388657
WAY-388657 is a Notum Pectinacetylesterase inhibitor with IC50 < 0.025 M.
ţT60057 أй½
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TP1545L1FFAGLDD amine saltFFAGLDD amine salt
FFAGLDD amine salt is MMP9 selective cleavage peptides, which used for cytosolic delivery of Doxorubi-cin (DOX) and achieve temporally and spatially controlled slow drug delivery and release.
ţTP1545L1 أй½
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T40652Meclizine
Meclizine (Meclozine) shows antihistamine activity and reversibly inhibits the interaction of histamine at the H1 receptors . Meclizine is a member of the piperazine class of H1 antagonists. Meclizine is an effective anti-motion sickness agent. Meclizine crosses the bloodCbrain barrier. Meclizine is an agonist ligand for mouse constitutive androstane receptor (CAR) and an inverse agonist for Human CAR. Meclizine can be used for the research of polyQ toxicity disorders, such as Huntington´s
ţT40652 أй½
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T8222SelpercatinibFVB/NRj mice,RET (WT),inhibit,Inhibitor,RET (G810R),LOXO 292,LOXO292,RET (V804M),Selper
Selpercatinib is a tyrosine kinase inhibitor with antineoplastic properties(IC50 of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M) , and RET (G810R), respectively)
ţT8222 أй½
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Fr13877Compound Fr13877Compound Fr13877
ţFr13877 أй½
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TN6982Diethyl phthalate
Diethyl phthalate is a endocrine disrupter affecting the apoptotic system in PC12 cells. Diethyl phthalate is widely used in many plastics and personal care products.
ţTN6982 أй½
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T7083GLPG1837GLPG-1837,ABBV 974,Cystic fibrosis transmembrane conductance regulator,Inhibitor,CFTR,Autoph
GLPG1837 is an effective CFTR potentiator, with EC50s of 3 nM and 339 nM for F508del and G551D CFTR, respectively.
ţT7083 أй½
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T7974Lynestrenolinhibit,progesteronelike,Pregnane,Inhibitor,immunostimulatory,zfPXR,Lynestrenol,PXR,hPXR
Lynestrenol is a synthetic progestational hormone, is the progesterone receptor agonist
ţT7974 أй½
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T6507Gabapentin hydrochlorideInhibitor,Gabapentin hydrochloride,Gabapentin,Calcium Channel,Ca channels,in
Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
ţT6507 أй½
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T38163ML-148ML-148,ML 148,selective,Inhibitor,prostaglandin-signaling,15-PGDH,15-Hydroxyprostaglandin dehy
ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM). ML-148 can be used to profile across a panel of related dehydrogenase or reductase enzymes and in studies about prostaglandin-signaling pathways.
ţT38163 أй½
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T6648Rotundine5-hydroxytryptamine Receptor,Inhibitor,Dopamine Receptor,Rotundine,5-HT Receptor,inhibit,Se
Rotundine (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.
ţT6648 أй½
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T60199NCRW0005-F05NCRW0005F05
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 value of 0.21 M. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson´s disease [1].
ţT60199 أй½
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T7712LDisomotide TFA 181477-43-0(free base)Disomotide TFA 181477430(free base),Disomotide TFA 181477 43 0(
Disomotide is an oligopeptide for the treatment of melanoma.
ţT7712L أй½
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T6874Lercanidipine hydrochlorideantihypertensive,Inhibitor,calcium,Lercanidipine,Lercanidipine hydrochlor
Lercanidipine is a calcium channel blocker of the dihydropyridine class.
ţT6874 أй½
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T6683STF-62247renal,STF-62247,VHL,carcinoma,inhibit,cytotoxic,cell,RCC,Inhibitor,STF62247,intracytoplasmi
STF-62247 is TGN inhibitor with IC50 of 0.625 M and 16 M in RCC4 and RCC4/VHL cells, respectively.
ţT6683 أй½