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T38332Complement factor D-IN-2；化合物Complement factor D-IN-2Complement factor D-IN-2
Complement factor D-IN-2 is an inhibitor of Complement factor D and reduces the excessive activation of complement factor D.
价 格：￥电议型 号：T38332产 地：中国大陆
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T38223N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide；N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamideN-(1-(3
N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide binds to the cannabinoid 1 (CB1) receptor with a Ki value of 365 nM in a radioligand binding assay using rat brain homogenate. It has an EC50 value of 698 nM for the peroxisome proliferator-activated receptor α (PPARα) in a luciferase reporter assay and, in rats, it decreases food intake. It does not inhibit fatty acid amide hydrolase (FAAH).
价 格：￥电议型 号：T38223产 地：中国大陆
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T38072HSGN-218；HSGN-218HSGN-218
HSGN-218 is a gut-restrictive antibiotic.1It is active againstC. difficile(MIC = 0.007 μg/ml) and clinical isolates ofC. difficile(MICs = 0.003-0.03 μg/ml) and is not cytotoxic to Caco-2 cells when used at concentrations ranging from 4 to 64 μg/ml. HSGN-218 (50 mg/kg) increases survival and protects mice fromC. difficilerecurrence in mouse models ofC. difficileinfection.
价 格：￥电议型 号：T38072产 地：中国大陆
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T378841,3-Linolein-2-Olein；1,3亚油酸-2-油酸甘油酯1,3-Linolein-2-Olein
1,3-Dilinoleoyl-2-oleoyl-rac-glycerol is a triacylglycerol that contains linoleic acid at the sn-1 and sn-3 positions and oleic acid at the sn-2 position. It has been found in grape seed, pumpkin seed, soybean, sunflower, and wheat germ oils, with the highest content in grape seed oil.
价 格：￥电议型 号：T37884产 地：中国大陆
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T3780Oroxin B；木蝴蝶苷BHypocretin-2；Hypocretin-2|||木蝴蝶苷B
Oroxin B (Hypocretin-2) has antioxidant activity.
价 格：￥电议型 号：T3780产 地：中国大陆
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T37095Quin-2 (potassium salt)；Quin-2 (potassium salt)Quin-2 (potassium salt)
Quin-2 is a high-affinity fluorescent calcium indicator (Kd = 115 nM for calcium). It displays high selectivity for calcium, as it is not affected by sodium gradients, membrane potential, or intracellular pH. High affinity probes like quin-2 are ideal for monitoring low levels of calcium, as are found in resting cells. Loadings of up to 2 mM quin-2 are without serious toxic effects, so quin-2 may be used to buffer intracellular calcium transients. Excitation/emission maxima for quin-2 are 339 an
价 格：￥电议型 号：T37095产 地：中国大陆
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T37020Endosidin-2；化合物Endosidin-2ES2|||Endosidin 2；ES2|||Endosidin 2
Endosidin-2 is an exocyst inhibitor, a cell-permeable benzylidene benzoylhydrazine, that binds to the exocyst component of the 70 kDa (EXO70) subunit of the exocyst complex (Kd = 253 μM, EXO70A1).Endosidin-2 disrupts protein translocation between the endosomes and plasma membrane, thereby facilitating translocation of proteins to the vesicle for degradation. It also inhibits recirculation of endocytosed transferrin to the plasma membrane in HeLa cells and targets multiple isoforms of mammalian E
价 格：￥电议型 号：T37020产 地：中国大陆
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T36968ARN-21934；化合物ARN-21934ARN-21934
ARN-21934 is a potent and selective inhibitor for human topoisomerase II α and topoisomerase II β. ARN-21934(IC50 = 2 μM) inhibits DNA relaxation as compared to the anticancer agent Etoposide (IC50=120 μM).
价 格：￥电议型 号：T36968产 地：中国大陆
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T36923CXCR2-IN-2CXCR2-IN-2CXCR2-IN-2
CXCR2-IN-2 is a selective CXCR2 antagonist that is brain penetrant and orally bioavailable, with IC50 values of 5.2 nM and 1 nM in the β-arrestin assay and CXCR2 Tango assay, respectively. It exhibits approximately 730-fold selectivity over CXCR1 and greater than 1900-fold selectivity over all other chemokine receptors. Furthermore, CXCR2-IN-2 effectively inhibits Gro-α induced CD11b expression in human whole blood, displaying an IC50 of 0.04 μM[1].
价 格：￥电议型 号：T36923产 地：中国大陆
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T36832PDE4B-IN-2；化合物PDE4B-IN-2A 33；A 33
PDE4B-IN-2 (A 33) is an orally active and selective PDE4B inhibitor with an IC50 of 15 nM. PDE4B-IN-2 inhibits PDE4D (IC50=1.7 ?M). PDE4B-IN-2 exhibits potent anti-inflammatory effects.
价 格：￥电议型 号：T36832产 地：中国大陆
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T36820Fluphenazine-N-2-chloroethane (hydrochloride)；Fluphenazine-N-2-chloroethane (hydrochloride)Fluphenaz
Fluphenazine is a traditional antipsychotic compound that tightly binds the dopamine D2 receptor (Ki = 0.55 nM) and also reversibly inhibits calmodulin at micromolar concentrations. Fluphenazine-N-2-chloroethane is a derivative of fluphenazine that contains an alkylating chlorethylamine chain, which produces irreversible protein binding. It is a relatively selective, irreversible antagonist of D2 receptors both in vitro (IC50 = 100 nM) and in vivo, inactivating approximately 90% of D2 receptors
价 格：￥电议型 号：T36820产 地：中国大陆
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T36782TAK1-IN-2；TAK1-IN-2TAK1-IN-2；TAK1-IN-2
TAK1-IN-2 is a potent and selective TAK1 inhibitor, with an IC50> of 2 nM[1].
价 格：￥电议型 号：T36782产 地：中国大陆
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T3671Vitexin-2"-O-rhamnoside；牡荆素鼠李糖苷Vitexin2"Orhamnoside|||inhibit|||牡荆素鼠李糖苷|||Vitexin-2''-O-rhamnoside||
Vitexin-2"-O-rhamnoside (Apigenin-8-C-glucoside) is a compound contributes to the protection against H O -mediated oxidative stress damage.
价 格：￥电议型 号：T3671产 地：中国大陆
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T3661Citarinostat；化合物CitarinostatACY241|||HDAC-IN-2；ACY241|||HDAC-IN-2
ACY-241, also known as Citarinostat (ACY241), is a potent, selective and orally available histone deacetylase (HDAC) inhibitor, with potential antineoplastic activity. Upon oral administration, ACY-241 inhibits the activity of HDACs; this results in an accumulation of highly acetylated chromatin histones, the induction of chromatin remodeling and an altered pattern of gene expression. This leads to the inhibition of tumor oncogene transcription, and the selective transcription of tumor suppresso
价 格：￥电议型 号：T3661产 地：中国大陆
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T36465Caylin-2；Caylin-2Caylin-2
Nutlin-3 is an activator of p53 that functions by inhibiting the interaction of p53 with MDM2, a negative regulator of p53 activity. Caylin-2 is a nutlin-3 analog in which trifluoromethyl groups have been substituted for chlorine on the 2 phenyl rings. At high concentrations, caylin-2 inhibits the growth of HCT116 cells with an IC50 of approximately 8 μM, making it about 10-fold less potent than nutlin-3. Interestingly, at concentrations between 5-100 nM, caylin-2 promotes the growth of HCT116 c
价 格：￥电议型 号：T36465产 地：中国大陆
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T36443(R,R)-CXCR2-IN-2(R,R)-CXCR2-IN-2(R,R)-CXCR2-IN-2
(R,R)-CXCR2-IN-2, a diastereoisomer of CXCR2-IN-2 (compound 68), functions as a brain-penetrant CXCR2 antagonist. It exhibits a pIC50 of 9 in the Tango assay and 6.8 in the HWB Gro-α induced CD11b expression assay[1].
价 格：￥电议型 号：T36443产 地：中国大陆
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T36097TNF-α-IN-2；TNF-α-IN-2TNF-α-IN-2
TNF-α-IN-2 is a highly potent and orally bioavailable inhibitor of tumor necrosis factor alpha (TNFα), exhibiting an IC50 of 25 nM in the HTRF assay. It exerts its inhibitory effects by inducing conformational changes in the TNFα trimer upon binding, resulting in disrupted signaling when the trimer interacts with TNFR1. TNF-α-IN-2 holds promise as a valuable tool for investigating the pathogenesis of rheumatoid arthritis[1].
价 格：￥电议型 号：T36097产 地：中国大陆
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T36087PI3K-IN-22；CAY10626CAY10626；CAY10626
PI3K-IN-22 is a dual kinase inhibitor of PI3Kα and mTOR, with IC50s of 0.9 and 0.6 nM respectively. PI3K-IN-22 could be used in cancer.
价 格：￥电议型 号：T36087产 地：中国大陆
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T35868BCAT-IN-2；BCAT 抑制剂2BCAT-IN-2
BCAT-IN-2 is an orally active and selective inhibitor of mitochondrial branched-chain aminotransferase (BCATm), inhibits BCATm and BCATc, and is used in obesity and dyslipidemia.
价 格：￥电议型 号：T35868产 地：中国大陆
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T357022-Heptanol；2-庚醇s-Heptyl alcohol|||Heptan-2-ol|||Heptanol-2；s-Heptyl alcohol|||Heptan-2-ol|||Heptanol
2-Heptanol (s-Heptyl alcohol) is a chemical compound found in the essential oil extracted from the rhizome of Curcuma angustifolia and Curcuma zedoaria. The rhizome essential oil demonstrates noteworthy antimicrobial and antioxidant properties.
价 格：￥电议型 号：T35702产 地：中国大陆
