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T5698TRPM8 antagonist 2TRPM8 antagonist 2
TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist, with an IC50 of 0.2 nM, used in the research of neuropathic pain syndromes.
价 格：￥电议型 号：T5698产 地：美洲
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T5829H4 Receptor antagonist 1H4 Receptor antagonist 1
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
价 格：￥电议型 号：T5829产 地：美洲
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T5962N-Ethyl-p-menthane-3-carboxamideN-Ethyl-p-menthane-3-carboxamide,TRPM8 antagonist WS-3,Cyclohexaneca
N-Ethyl-p-menthane-3-carboxamide is an agonist of TRPM8( EC50 : 3.7 μM).
价 格：￥电议型 号：T5962产 地：美洲
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T8649TMBIM6 antagonist-1；1-（2-氨基苯基）-3-（3-硝基苯基）-2-丙烯-1-酮BAX-inhibitor-1|||BIA；BAX-inhibitor-1|||1-（2-氨基苯基）
TMBIM6 antagonist-1 (BAX-inhibitor-1) is a bax inhibitor
价 格：￥电议型 号：T8649产 地：中国大陆
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T84384i；化合物4iCHEMBL1269981|||5-HT3 antagonist-4i；CHEMBL1269981|||5-HT3 antagonist-4i
4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.
价 格：￥电议型 号：T8438产 地：中国大陆
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T83972NOX-6-18；化合物 NOX-6-18GPR132 antagonist 1|||GPR132-B-160；GPR132 antagonist 1|||GPR132-B-160
NOX-6-18 (GPR132-B-160) is a highly potent and selective GPR132 antagonist with insulinotropic activity that modulates macrophage reprogramming in pancreatic islets and reduces weight gain.
价 格：￥电议型 号：T83972产 地：中国大陆
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T83779EP4 Antagonist 14；化合物 EP4 Antagonist 14Prostaglandin E2 Receptor 4 Antagonist 14|||PGE2 Receptor 4 A
EP4 antagonist 14 is a prostaglandin E2 receptor subtype EP4 antagonist, demonstrating an IC50 of 1.1 nM in a HEK293 human receptor reporter assay and blocking β-arrestin recruitment due to PGE2 with an IC50 of 0.9 nM. At 10 ?M, it reduces PGE2-stimulated mRNA levels of Il-4, macrophage mannose receptor 1 (Mrc1), chitinase-like protein 3 (Chil3), chemokine (C-X-C) motif ligand 1 (Cxcl1), triggering receptor expressed on myeloid cells 2 (Trem2), and arginase-1 (Arg1) in RAW 264.7 macrophages. Whe
价 格：￥电议型 号：T83779产 地：中国大陆
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T832895-HT6R antagonist 2；化合物 5-HT6R antagonist 25-HT6R antagonist 2
Compound 29 is a 5-HT6R antagonist that acts by inhibiting the 5-HT6 receptor.
价 格：￥电议型 号：T83289产 地：中国大陆
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T83119Androgen receptor antagonist 9；化合物 Androgen receptor antagonist 9Androgen receptor antagonist 9
Androgen Receptor Antagonist 9 (compound 28) serves as an antagonist to the androgen receptor [1].
价 格：￥电议型 号：T83119产 地：中国大陆
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T82797C5aR1 antagonist peptide；化合物 C5aR1 antagonist peptideC5aR1 antagonist peptide
C5aR1 antagonist peptide, a biologically active linear peptide originating from the C-terminus of the chemokine complement fragment 5 anaphylatoxin (C5a), inhibits C5a binding and activity at human and rat C5a receptors. Overexpression of C5a is linked to various immunoinflammatory diseases, including arthritis, Alzheimer’s disease, cystic fibrosis, and systemic lupus erythematosus.
价 格：￥电议型 号：T82797产 地：中国大陆
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T82772CB2 receptor antagonist 2；化合物 CB2 receptor antagonist 2CB2 receptor antagonist 2
Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 μM. It engages in strong interactions with residues L17, W6.48, V6.51, and C7.42 [1].
价 格：￥电议型 号：T82772产 地：中国大陆
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T82703CMKLR1 antagonist 1；化合物 CMKLR1 antagonist 1CMKLR1 antagonist 1
CMKLR1 antagonist 1 (compound S-26d) is a potent, orally active antagonist of the chemokine-like receptor 1 (CMKLR1), exhibiting a pIC50 of 7.44 in hCMKLR1-transfected CHO cells. It is applicable in the research of psoriasis and metabolic diseases [1].
价 格：￥电议型 号：T82703产 地：中国大陆
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T82605DB21, Galectin-1 Antagonist；化合物 DB21, Galectin-1 AntagonistDB21, Galectin-1 Antagonist
DB21, Galectin-1 Antagonist, is a peptidomimetic conjugated with dibenzofuran, serving as an allosteric inhibitor of galectin-1 (GAL1) interactions with glycans on cell surfaces. This compound enhances the inhibition of angiogenesis and tumor growth in melanoma, lung adenocarcinoma, and ovarian cancer models [1].
价 格：￥电议型 号：T82605产 地：中国大陆
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T82357GABA receptor Antagonist 1；化合物 GABA receptor Antagonist 1GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P. xylostella, S. frugiperda, S. exigua, and S. litura with respective LC50 values of 0.09, 0.84, 0.87, and 0.68 mg/L. Moreover, this compound exhibits moderate toxicity to honeybees (48 h, ID50 = 2.22 μg/adult) and low toxicity to zebrafish (LC50: 42.4 mg/L) [1].
价 格：￥电议型 号：T82357产 地：中国大陆
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T82264GPR34 receptor antagonist 3；化合物 GPR34 receptor antagonist 3GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner, demonstrating an IC50 value of 0.680 μM without significant cytotoxicity. Additionally, it displays antisensory activity in a mouse neuropathic pain model [1].
价 格：￥电议型 号：T82264产 地：中国大陆
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T82020J5 peptide；化合物 J5 peptideMyelin basic protein (85-99) antagonist；Myelin basic protein (85-99) antago
J5 peptide, an MBP inhibitor, competitively inhibits the binding of MBP 85-99 to HLA-DR2, and mitigates PLP 139-151/MBP 85-99-induced experimental autoimmune encephalomyelitis (EAE) in mice. It is utilized in research pertaining to inflammatory and immune diseases [1].
价 格：￥电议型 号：T82020产 地：中国大陆
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T81888mAChR antagonist 1；化合物 mAChR antagonist 1mAChR antagonist 1
Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes, respectively [1].
价 格：￥电议型 号：T81888产 地：中国大陆
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T81801mGluR5 antagonist-1；化合物 mGluR5 antagonist-1mGluR5 antagonist-1
mGluR5 antagonist-1 (compound 10) is a potent mGluR5 inhibitor exhibiting an IC50 of 11.5 nM and demonstrates antidepressant effects [1].
价 格：￥电议型 号：T81801产 地：中国大陆
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T81579P2X7 receptor antagonist-4；化合物 P2X7 receptor antagonist-4P2X7 receptor antagonist-4
Compound 14a (P2X7 receptor antagonist-4) is a P2X7R antagonist with IC50 values of 64.7 nM in humans and 10.1 nM in mice. It inhibits the activation of the NLRP3 inflammasome, which subsequently reduces the expression of caspase-1, gasdermin D, IL-1β, and IL-18 in the kidneys of mice with sepsis-induced damage [1].
价 格：￥电议型 号：T81579产 地：中国大陆
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T79793CRF1 receptor antagonist-1；化合物 CRF1 receptor antagonist-1CRF1 receptor antagonist-1
CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to congenital adrenal hyperplasia (CAH) [1].
价 格：￥电议型 号：T79793产 地：中国大陆
