T5393CK1-IN-1PUN51207

CK1-IN-1, compound 1c reported in patent WO2015119579A1, is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.

价 格：￥电议型 号：T5393产 地：中国大陆

T5184ERK5-IN-1

ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM). It also inhibits LRRK2[G2019S] (IC50: 26 nM).

价 格：￥电议型 号：T5184产 地：中国大陆

T5093Pim1/AKK1-IN-1LKB1/AAK1 dual inhibitor；MDK-2275

Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK.

价 格：￥电议型 号：T5093产 地：中国大陆

T4642Tenovin-2

价 格：￥电议型 号：T4642产 地：中国大陆

T4438Porcn-IN-1Porcupine-IN-1

Porcupine-IN-1 is an effective porcupine inhibitor (IC50: 0.5±0.2 nM).

价 格：￥电议型 号：T4438产 地：中国大陆

T4376Nampt-IN-1LSN3154567

Nampt-IN-1 (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM.

价 格：￥电议型 号：T4376产 地：中国大陆

T4365FL-411FL411；FL 411；BRD4-IN-1

FL-411 is a potent and selective BRD4 inhibitor with an IC50 of 0.43±0.09 μM for BRD4.

价 格：￥电议型 号：T4365产 地：中国大陆

T4332c-Kit-IN-1PDGFR inhibitor 1；DCC-2618

DCC-2618 is an effective inhibitor of c-Met and c-Kit (IC50s<200 nM).

价 格：￥电议型 号：T4332产 地：中国大陆

T4328OSS_128167SIRT6-IN-1

OSS_128167 is a specific SIRT6 inhibitor, and for SIRT6(IC50=89 μM), SIRT1(IC50=1578 μM) and SIRT2(IC50=751 μM).

价 格：￥电议型 号：T4328产 地：中国大陆

T4288hVEGF-IN-1

hVEGF-IN-1 inhibits human VEGF-A translation and has antitumor activity.

价 格：￥电议型 号：T4288产 地：中国大陆

T4256PTP1B-IN-2

PTP1B-IN-2 is an effective protein tyrosine phosphatase 1B (PTP1B) inhibitor(IC50=50 nM).

价 格：￥电议型 号：T4256产 地：中国大陆

T4231MD2-IN-1

MD2-IN-1 is an inhibitor of Myeloid differentiation protein 2 (MD2) with a KD of 189 μM for the recombinant human MD2 (rhMD2).

价 格：￥电议型 号：T4231产 地：中国大陆

T4223MitapivatPKR-IN-1

Mitapivat, also known as PKM2 activator 1020 is a PKM2 activator (pyruvate kinase activator) for the treatment of pyruvate kinase deficiency.

价 格：￥电议型 号：T4223产 地：中国大陆

T4214KDM4D-IN-1

KDM4D-IN-1 is a KDM4D inhibitor (IC50: 0.41±0.03 μM).

价 格：￥电议型 号：T4214产 地：中国大陆

T4142PCC0208009IDO-IN-2；DO-IN-2；IDO inhibitor 1

IDO-IN-2 is an IDO inhibitor extracted from patent WO/2015031295 A1, compound example 1.

价 格：￥电议型 号：T4142产 地：中国大陆

T4140IRAK4-IN-1

IRAK4-IN-1 is an interleukin-1 receptor associated kinase 4 (IRAK4) inhibitor with an IC50 of 7 nM.

价 格：￥电议型 号：T4140产 地：中国大陆

T4075Sulfatinib索凡替尼；KDR-IN-1

Sulfatinib may be a potent drug for cancer. It inhibits KDR and FGFR1 enzymatic activity. It also is a hERG inhibitor.

价 格：￥电议型 号：T4075产 地：中国大陆

T4044DprE1-IN-2

DprE1-IN-2 is an effective DprE1 inhibitor.

价 格：￥电议型 号：T4044产 地：中国大陆

T40242DEPTOR-IN-1

DEPTOR-IN-1 is an inhibitor of DEPTOR with a Kd of 9.3 μM.

价 格：￥电议型 号：T40242产 地：中国大陆

T39669TLR7/8/9-IN-1TLR7/8/9-IN-1

TLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.

价 格：￥电议型 号：T39669产 地：中国大陆