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T82605DB21, Galectin-1 Antagonist；化合物 DB21, Galectin-1 AntagonistDB21, Galectin-1 Antagonist
DB21, Galectin-1 Antagonist, is a peptidomimetic conjugated with dibenzofuran, serving as an allosteric inhibitor of galectin-1 (GAL1) interactions with glycans on cell surfaces. This compound enhances the inhibition of angiogenesis and tumor growth in melanoma, lung adenocarcinoma, and ovarian cancer models [1].
价 格：￥电议型 号：T82605产 地：中国大陆
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T82455Epoetin beta；化合物 Epoetin betaGenetical recombination|||rhEPO|||EPOCH；Genetical recombination|||rhEPO
Epoetin beta (rhEPO), a recombinant erythropoietin, is crucial for sustaining erythropoiesis and is utilized in anemia research [1].
价 格：￥电议型 号：T82455产 地：中国大陆
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T82357GABA receptor Antagonist 1；化合物 GABA receptor Antagonist 1GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P. xylostella, S. frugiperda, S. exigua, and S. litura with respective LC50 values of 0.09, 0.84, 0.87, and 0.68 mg/L. Moreover, this compound exhibits moderate toxicity to honeybees (48 h, ID50 = 2.22 μg/adult) and low toxicity to zebrafish (LC50: 42.4 mg/L) [1].
价 格：￥电议型 号：T82357产 地：中国大陆
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T82264GPR34 receptor antagonist 3；化合物 GPR34 receptor antagonist 3GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner, demonstrating an IC50 value of 0.680 μM without significant cytotoxicity. Additionally, it displays antisensory activity in a mouse neuropathic pain model [1].
价 格：￥电议型 号：T82264产 地：中国大陆
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T82020J5 peptide；化合物 J5 peptideMyelin basic protein (85-99) antagonist；Myelin basic protein (85-99) antago
J5 peptide, an MBP inhibitor, competitively inhibits the binding of MBP 85-99 to HLA-DR2, and mitigates PLP 139-151/MBP 85-99-induced experimental autoimmune encephalomyelitis (EAE) in mice. It is utilized in research pertaining to inflammatory and immune diseases [1].
价 格：￥电议型 号：T82020产 地：中国大陆
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T81888mAChR antagonist 1；化合物 mAChR antagonist 1mAChR antagonist 1
Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes, respectively [1].
价 格：￥电议型 号：T81888产 地：中国大陆
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T81835MC-betaglucuronide-MMAE-2；化合物 MC-betaglucuronide-MMAE-2MC-betaglucuronide-MMAE-2
MC-betaglucuronide-MMAE-2 is an ADC (antibody-drug conjugate) agent-linker conjugate that exhibits potent antitumor activity; it consists of MMAE (a tubulin polymerization inhibitor) connected through the cleavable linker MC-betaglucuronide.
价 格：￥电议型 号：T81835产 地：中国大陆
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T81801mGluR5 antagonist-1；化合物 mGluR5 antagonist-1mGluR5 antagonist-1
mGluR5 antagonist-1 (compound 10) is a potent mGluR5 inhibitor exhibiting an IC50 of 11.5 nM and demonstrates antidepressant effects [1].
价 格：￥电议型 号：T81801产 地：中国大陆
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T8178Acetagastrodin；乙酰天麻素Acegastrodine；乙酰天麻素|||Acegastrodine
Acetagastrodin (Acegastrodine) has an antispasmodic effect on vascular smooth muscle.
价 格：￥电议型 号：T8178产 地：中国大陆
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T81579P2X7 receptor antagonist-4；化合物 P2X7 receptor antagonist-4P2X7 receptor antagonist-4
Compound 14a (P2X7 receptor antagonist-4) is a P2X7R antagonist with IC50 values of 64.7 nM in humans and 10.1 nM in mice. It inhibits the activation of the NLRP3 inflammasome, which subsequently reduces the expression of caspase-1, gasdermin D, IL-1β, and IL-18 in the kidneys of mice with sepsis-induced damage [1].
价 格：￥电议型 号：T81579产 地：中国大陆
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T8114Quercetagetin；栎草亭6-Hydroxyquercetin；栎草亭|||6-Hydroxyquercetin
Quercetagetin (6-Hydroxyquercetin) (6-Hydroxyquercetin) is the major flavonoid isolated from Citrus unshiu. It is a moderately potent and selective, cell-permeable pim-1 kinase inhibitor (IC50: 0.34 μM).
价 格：￥电议型 号：T8114产 地：中国大陆
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T80851VSTx-3；化合物 VSTx-3Kappa-TRTX-Gr4a|||κ-Theraphotoxin-Gr4a|||Voltage sensor toxin 3|||Peptide F；Kappa-T
VSTx-3 is a potassium voltage-gated channel (K_V) blocker, which has also been shown to be a potent tetrodotoxin-sensitive (TTX-sensitive) sodium channel inhibitor, with particular efficacy against NaV1.8 channels, as evidenced by its half-maximal inhibitory concentration (IC_50) values of 0.19 μM for hNaV1.3, 0.43 μM for hNaV1.7, and 0.77 μM for hNaV1.8 channels.
价 格：￥电议型 号：T80851产 地：中国大陆
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T79793CRF1 receptor antagonist-1；化合物 CRF1 receptor antagonist-1CRF1 receptor antagonist-1
CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to congenital adrenal hyperplasia (CAH) [1].
价 格：￥电议型 号：T79793产 地：中国大陆
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T79786H4R antagonist 2；化合物 H4R antagonist 2H4R antagonist 2
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid arthritis [1] (page 68).
价 格：￥电议型 号：T79786产 地：中国大陆
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T79782FPR1 antagonist 2；化合物 FPR1 antagonist 2FPR1 antagonist 2
Compound 25b, an FPR1 antagonist, exhibits potent inhibition of the formyl peptide receptor 1 with an IC50 of 70 nM. It concurrently hampers cell proliferation and triggers apoptosis, diminishing cell growth and migration, yet paradoxically augments angiogenesis [1].
价 格：￥电议型 号：T79782产 地：中国大陆
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T79781FPR1 antagonist 1；化合物 FPR1 antagonist 1FPR1 antagonist 1
Compound 24a, an FPR1 antagonist, demonstrates potent inhibition of the formyl peptide receptor 1 (FPR1) with an IC50 value of 25 nM. It impedes cell proliferation and promotes apoptosis, thereby inhibiting cell growth. This compound also attenuates cell migration and concurrently promotes angiogenesis [1].
价 格：￥电议型 号：T79781产 地：中国大陆
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T79772RARα antagonist 1；化合物 RARα antagonist 1RARα antagonist 1
Compound 21, an orally active and selective RARα antagonist, exhibits a potent inhibition of the retinoic acid receptor α with an IC50 of 4.6 nM [1].
价 格：￥电议型 号：T79772产 地：中国大陆
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T796845-HT6R antagonist 1；化合物 5-HT6R antagonist 15-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability but also reverses MK-801-induced memory impairments in rats, suggesting its utility in Alzheimer´s disease (AD) research [1].
价 格：￥电议型 号：T79684产 地：中国大陆
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T79575ET receptor antagonist 3；化合物 ET receptor antagonist 3ET receptor antagonist 3
"ET receptor antagonist 3 (compound 17d) is an orally active ET receptor antagonist with an IC50 of 0.26 nM, utilized for pulmonary arterial hypertension (PAH) research. This compound demonstrates efficacy in mitigating monocrotaline-induced PAH in a rat model [1]."
价 格：￥电议型 号：T79575产 地：中国大陆
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T79574ET receptor antagonist 2；化合物 ET receptor antagonist 2ET receptor antagonist 2
ET Receptor Antagonist 2 (Compound 16j) is an orally active ET receptor antagonist with an IC50 of 0.22 nM, suitable for pulmonary arterial hypertension (PAH) research. It has been shown to mitigate monocrotaline-induced PAH in a rat model [1].
价 格：￥电议型 号：T79574产 地：中国大陆
