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  • T78939AChE-IN-31；化合物 AChE-IN-31AChE-IN-31

    AChE-IN-31 (compound 1), a non-competitive acetylcholinesterase (AChE) inhibitor, exhibits potential for Alzheimer´s disease research [1].

    价 格：￥电议型 号：T78939产 地：中国大陆

  • T78927PSMA-IN-3；化合物 PSMA-IN-3PSMA-IN-3

    PSMA-IN-3 (compound 17) is a novel, high-affinity inhibitor of Prostate-Specific Membrane Antigen (PSMA) with an inhibitory concentration (IC50) of 13 nM, showing potential for the development of an 18F-labeled radioligand for positron emission tomography (PET) imaging of PSMA in prostate cancer [1].

    价 格：￥电议型 号：T78927产 地：中国大陆

  • T78906CDK/HDAC-IN-3；化合物 CDK/HDAC-IN-3CDK/HDAC-IN-3

    CDK/HDAC-IN-3 is an orally active dual inhibitor of HDACs and CDKs, offering potent and selective inhibition of CDK9, CDK12, CDK13, HDAC1, HDAC2, and HDAC3, with IC50 values of 98.32 nM, 98.85 nM, 100 nM, 62.12 nM, 93.28 nM, and 82.87 nM, respectively. This compound is applicable in the treatment of acute myeloid leukemia (AML) [1].

    价 格：￥电议型 号：T78906产 地：中国大陆

  • T78881α-Glucosidase-IN-36；化合物 α-Glucosidase-IN-36α-Glucosidase-IN-36

    α-Glucosidase-IN-36 (compound 5g) is a potent inhibitor of α-glucosidase, exhibiting an IC50 value of 6.69 ± 0.18 μM and inhibition constants Ki and Kis of 1.65 μM and 4.54 μM, respectively. It is hypothesized to suppress α-glucosidase activity by interacting with its active site and altering the enzyme´s secondary structure. The compound is relevant for use in research on type 2 diabetes mellitus (T2DM) [1].

    价 格：￥电议型 号：T78881产 地：中国大陆

  • T78880Tubulin/HDAC-IN-3；化合物 Tubulin/HDAC-IN-3Tubulin/HDAC-IN-3

    Tubulin/HDAC-IN-3 (compound 12a) serves as a potent dual inhibitor of tubulin polymerization and HDAC1/8, exhibiting IC50 values of 5.4 μM for tubulin polymerization, and 0.155 and 0.177 μM for HDAC1 and HDAC8, respectively. Its mechanism of action includes obstructing the cell cycle, triggering apoptosis, and suppressing colony formation [1].

    价 格：￥电议型 号：T78880产 地：中国大陆

  • T78870TWIK-1/TREK-1-IN-3；TWIK-1/TREK-1抑制剂3TWIK-1/TREK-1-IN-3

    TWIK-1/TREK-1-IN-3 is a selective and potent inhibitor of potassium channel TREK-1, inhibiting TREK-1 homodimers and TWIK-1/TREK-1 heterodimers containing two-pore-domain potassium (K2p) channels.TWIK-1/TREK-1-IN-3 exhibits antidepressant activity and can be used in the study of depression.

    价 格：￥电议型 号：T78870产 地：中国大陆

  • T78865α-Glucosidase-IN-34；化合物 α-Glucosidase-IN-34α-Glucosidase-IN-34

    α-Glucosidase-IN-34 (compound 7f) is a potent inhibitor of α-glucosidase, exhibiting an IC50 of 2.90 μM, and is applicable in research related to type 2 diabetes and hyperglycemia [1].

    价 格：￥电议型 号：T78865产 地：中国大陆

  • T78864α-Glucosidase-IN-33；化合物 α-Glucosidase-IN-33α-Glucosidase-IN-33

    α-Glucosidase-IN-33 (compound 7c), with an IC50 of 2.39 μM, is a potent inhibitor of α-glucosidase and is relevant in research on type 2 diabetes and hyperglycemia [1].

    价 格：￥电议型 号：T78864产 地：中国大陆

  • T78852HPK1-IN-39；化合物 HPK1-IN-39HPK1-IN-39

    HPK1-IN-39 (Compound 10n), a selective inhibitor of Hematopoietic Progenitor Kinase 1 (HPK1) with an inhibitory concentration (IC50) of 29 nM, impedes the phosphorylation of SLP76. This compound is applicable in the research of cancer immunotherapy [1].

    价 格：￥电议型 号：T78852产 地：中国大陆

  • T78850EGFR/BRAFV600E-IN-3；化合物 EGFR/BRAFV600E-IN-3EGFR/BRAFV600E-IN-3

    EGFR/BRAFV600E-IN-3 is an inhibitor targeting EGFR, BRAFV600E, and EGFRT790M with IC50 values of 57 nM, 68 nM, and 9.70 nM, respectively. It induces apoptosis and exhibits promising antioxidant activity [1].

    价 格：￥电议型 号：T78850产 地：中国大陆

  • T78848MAO-IN-3；化合物 MAO-IN-3MAO-IN-3

    MAO-IN-3 (Compound 5), a reversible and competitive monoamine oxidase (MAO) inhibitor with inhibition constants (K i) of 0.6 μM for MAO A and 0.2 μM for MAO B, effectively suppresses LN-229 glioblastoma cell proliferation, as denoted by an inhibitory concentration (IC50) of 0.8 μM. This compound holds potential application in cancer research [1].

    价 格：￥电议型 号：T78848产 地：中国大陆

  • T78841Nrf2-IN-3；化合物 Nrf2-IN-3Nrf2-IN-3

    Nrf2-IN-3 (Compound R16), a Nrf2 inhibitor, binds to KEAP1 mutants (G333C mKEAP1) thereby restoring the impaired KEAP1/NRF2 interactions. This restoration sensitizes KEAP1-mutant cancer cells to chemotherapeutic agents, such as Cisplatin and Gefitinib, by reestablishing the functionality of the mKEAP1/NRF2 complex [1].

    价 格：￥电议型 号：T78841产 地：中国大陆

  • T78823Quorum Sensing-IN-3；Quorum Sensing抑制剂1QS-IN-1；QS-IN-1

    Quorum Sensing-IN-3 (QS-IN-1) is a compound with inhibitory effects on bacterial community sensing, which inhibits the exchange of information between bacteria and inhibits biofilm formation.

    价 格：￥电议型 号：T78823产 地：中国大陆

  • T78819VEGFR-2-IN-33；化合物 VEGFR-2-IN-33VEGFR-2-IN-33

    VEGFR-2-IN-33 (Compound 4d), a potent VEGFR inhibitor with an IC50 value of 61.04 nM, demonstrates significant inhibition of HepG2 cell proliferation, achieving an IC50 of 4.31 nM. This compound is utilized for hepatocellular carcinoma (HCC) research [1].

    价 格：￥电议型 号：T78819产 地：中国大陆

  • T78817AChE-IN-39；化合物 AChE-IN-39AChE-IN-39

    AChE-IN-39 (Compound 7c), with an IC50 value of 0.058 μM, is an acetylcholinesterase (AChE) inhibitor known for its DPPH scavenging activity and potential to ameliorate cognitive impairments in an aluminum chloride (AlCl3)-induced amnesia animal model, suggesting its usefulness in Alzheimer´s disease research [1].

    价 格：￥电议型 号：T78817产 地：中国大陆

  • T78815MOZ-IN-3；化合物 MOZ-IN-3MOZ-IN-3

    MOZ-IN-3 (Compound 6j), a potent KAT6A (MOZ) acetyltransferase inhibitor with an IC50 of 30 nM, exhibits antitumor activity against multiple myeloid leukemia cell lines, including HL-60, U937, SKNO-1, and K562. This compound also demonstrates favorable metabolic stability and pharmacokinetics [1].

    价 格：￥电议型 号：T78815产 地：中国大陆

  • T78812HBV-IN-36；化合物 HBV-IN-36HBV-IN-36

    HBV-IN-36 (also known as compound 42) is a hepatitis B virus (HBV) inhibitor with an IC50 of 2 μM, exhibiting anti-HBV activity characterized by an EC50 of 0.58 μM [1].

    价 格：￥电议型 号：T78812产 地：中国大陆

  • T78794α-Glucosidase-IN-31；化合物 α-Glucosidase-IN-31α-Glucosidase-IN-31

    α-Glucosidase-IN-31 (compound R1) is a potent oral α-Glucosidase inhibitor with an IC50 of 10.1 μM, demonstrating significant blood glucose reduction and antidiabetic activity [1].

    价 格：￥电议型 号：T78794产 地：中国大陆

  • T78786MmpL3-IN-3；化合物 MmpL3-IN-3MmpL3-IN-3

    MmpL3-IN-3 (Compound 12), an MmpL3 inhibitor, exhibits potent anti-tuberculosis activity with a minimum inhibitory concentration (MIC) of 0.1 μM against H37Rv and demonstrates good metabolic stability in mouse liver microsomes. This compound is valuable for anti-tubercular research [1].

    价 格：￥电议型 号：T78786产 地：中国大陆

  • T78784RIPK3-IN-3；化合物 RIPK3-IN-3RIPK3-IN-3

    RIPK3-IN-3 (compound 20) is a selective RIPK3 inhibitor that demonstrates potent activity with an IC50 value of 10 nM. This compound effectively blocks RIPK3-mediated phosphorylation of MLKL, preventing its oligomerization and subsequent induction of necroptosis. Additionally, RIPK3-IN-3 suppresses CXCL5 secretion and impedes AsPC-1 cell migration and invasion [1].

    价 格：￥电议型 号：T78784产 地：中国大陆

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