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T39798S1P2 antagonist 1；S1P2 antagonist 1S1P2 antagonist 1
S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.
价 格：￥电议型 号：T39798产 地：中国大陆
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T39762AHR antagonist 5 free base；化合物AHR antagonist 5 free baseAHR antagonist 5 free base
AHR antagonist 5 free base is an orally active antagonist of AHR with IC50s of ~35-150 nM in human and rodent cell lines.
价 格：￥电议型 号：T39762产 地：中国大陆
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T39742CXCR4 antagonist 2；CXCR4 antagonist 2CXCR4 antagonist 2
CXCR4 antagonist 2 is a CXCR4 antagonist with an IC 50 value of 47 nM.
价 格：￥电议型 号：T39742产 地：中国大陆
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T39662CCR4 antagonist 3 hydrochloride；CCR4 antagonist 3 hydrochlorideCCR4 antagonist 3 hydrochloride
CCR4 antagonist 3 hydrochloride is an orally active, potent and selective CCR4 antagonist. CCR4 antagonist 3, featuring a novel piperidinyl-azetidine motif, has IC 50 s of 22 nM and 50 nM in the calcium flux and CTX assay. CCR4 antagonist 3 has antitumor activity.
价 格：￥电议型 号：T39662产 地：中国大陆
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T39661CCR4 antagonist 3CCR4 antagonist 3CCR4 antagonist 3
CCR4 antagonist 3 is an orally active, potent and selective CCR4 antagonist. CCR4 antagonist 3, featuring a novel piperidinyl-azetidine motif, has IC 50 s of 22 nM and 50 nM in the calcium flux and CTX assay. CCR4 antagonist 3 has antitumor activity.
价 格：￥电议型 号：T39661产 地：中国大陆
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T39078CXCR7 antagonist-1；CXCR7拮抗剂1CXCR7 antagonist-1；CXCR7 antagonist-1
CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7. CXCR7 antagonist-1 prevents tumor cell proliferation and tumor formation and can be used in studies about inflammatory diseases.
价 格：￥电议型 号：T39078产 地：中国大陆
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T38910mGluR2 antagonist 1；mGluR2 antagonist 1mGluR2 antagonist 1
mGluR2 antagonist 1 is a potent and selective class of negative allosteric modulator targeting the metabotropic glutamate receptor 2 (mGluR2) with high oral bioavailability. It displays a remarkable affinity for mGluR2, with an IC50 value of 9 nM. Furthermore, it exhibits excellent permeability across the blood-brain barrier, making it a promising candidate for central nervous system-related studies or therapies.
价 格：￥电议型 号：T38910产 地：中国大陆
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T38634Histamine H4 receptor antagonist-1；Histamine H4 receptor antagonist-1Histamine H4 receptor antagonis
Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
价 格：￥电议型 号：T38634产 地：中国大陆
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T38622Bcl-xL antagonist 2；Bcl-xL拮抗剂2Bcl-xL antagonist 2
Bcl-xL antagonist 2 is an effective and selective antagonist of Bcl-xL with an IC50 of 91 nM and a Ki of 65 nM. Bcl-xL antagonist 2 induces apoptosis in cancer cells and can be used in studies about chronic lymphocytic leukemia and non-Hodgkin’s lymphoma.
价 格：￥电议型 号：T38622产 地：中国大陆
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T38595EP4 receptor antagonist 3EP4 receptor antagonist 3EP4 receptor antagonist 3
EP4 receptor antagonist 3 is a highly potent and specific inhibitor of the EP4 receptor. It is intended for research purposes in studying EP4 receptor-mediated diseases such as acute and chronic pain, osteoarthritis, rheumatoid arthritis, and cancer.
价 格：￥电议型 号：T38595产 地：中国大陆
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T38226TSHR antagonist S37b；TSHR antagonist S37bTSHR antagonist S37b
TSHR antagonist S37b, the less potent enantiomer of TSHR antagonist S37a, exhibits minimal efficacy in inhibiting the thyrotropin receptor (TSHR). It is utilized in thyroid function research[1].
价 格：￥电议型 号：T38226产 地：中国大陆
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T38139Orexin receptor antagonist 2；Orexin receptor antagonist 2Orexin receptor antagonist 2
Orexin Receptor Antagonist 2 (compound 30), characterized by its potent antagonistic activity with pKis of 7.69 and 9.78, holds promise for insomnia research[1].
价 格：￥电议型 号：T38139产 地：中国大陆
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T37793A2B receptor antagonist 2；化合物A2B receptor antagonist 2A2B receptor antagonist 2；A2B receptor antagon
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
价 格：￥电议型 号：T37793产 地：中国大陆
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T37792A2A receptor antagonist 1；化合物A2A receptor antagonist 1CPI-444 analog|||A2A receptor antagonist 1；CPI
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
价 格：￥电议型 号：T37792产 地：中国大陆
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T37429TRPV3 antagonist 74a；TRPV3 拮抗剂74aTRPV3 74a；TRPV3 74a
TRPV3 antagonist 74a (TRPV3 74a) is a specific TRPV3 antagonist for the study of neurological disorders.
价 格：￥电议型 号：T37429产 地：中国大陆
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T37223Glucagon Receptor Antagonist I；Glucagon Receptor Antagonist IGlucagon Receptor Antagonist I
Glucagon receptor antagonist I is a competitive antagonist of the glucagon receptor (GCGR; IC50 = 181 nM). It blocks glucagon-induced glycogenolysis in primary human hepatocytes and isolated liver. Glucagon receptor antagonist I, at 50 mg/kg, reduces the increase in glucose levels observed after intraperitoneal administration of glucagon in humanized mice. Glucagon receptor antagonist inactive control does not prevent glucagon-mediated actions.
价 格：￥电议型 号：T37223产 地：中国大陆
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T37003GnRH antagonist 2GnRH antagonist 2GnRH antagonist 2
GnRH antagonist 2 (formula I) is a potent GnRH receptor antagonist with valuable applications in endometriosis research[1].
价 格：￥电议型 号：T37003产 地：中国大陆
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T36982CXCR3 Antagonist 6cCXCR3 Antagonist 6cCXCR-3 Antagonist 6c|||CXCR3 Antagonist 6c
CXCR3 antagonist 6c is an antagonist of chemokine (C-X-C motif) receptor 3 (CXCR3).1It inhibits calcium mobilization induced by chemokine (C-X-C motif) ligand 11 (CXCL11) in HEK293 cells expressing the human receptor (IC50= 0.06 μM). It is selective for CXCR3 over a panel of 14 human G protein-coupled receptors at 10 μM. CXCR3 antagonist 6c inhibits CXCR3-mediated migration of isolated human T cells (IC50= ~100 nM).
价 格：￥电议型 号：T36982产 地：中国大陆
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T3680ISO-1；化合物ISO1MIF Antagonist|||ISO 1；MIF Antagonist|||ISO 1
ISO-1 (MIF Antagonist) is an inhibitor of the dopachrome tautomerase activity, blocks the activation of NF-κB and TNF-α secretion from LPS-treated macrophages.
价 格：￥电议型 号：T3680产 地：中国大陆
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T36744CDK9 Antagonist-1；CDK9 Antagonist-1CDK9 Antagonist-1；CDK9 Antagonist-1
CDK9 Antagonist-1 (compounds 11c) is a potent and selective CDK9 degrader based on PROTAC, with an IC50 of 17 μM in MCF-7 cell lines. Natural product Wogonin binds ubiquitin E3 ligase cereblon (CRBN) via a linker to form PROTAC[1].
价 格：￥电议型 号：T36744产 地：中国大陆
