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  • T61697GPVI antagonist 1；化合物 GPVI antagonist 1GPVI antagonist 1

    GPVI antagonist 1 (compound 5) functions as an antagonist for the glycoprotein VI (GPVI) platelet receptor. It effectively inhibits collagen-induced platelet aggregation, demonstrating an IC50 value of 25.3 μM [1].

    价 格：￥电议型 号：T61697产 地：中国大陆

  • T61650CXCR4 antagonist 9；化合物 CXCR4 antagonist 9CXCR4 antagonist 9

    CXCR4 antagonist 9 (Compound 2) is a potent CXCR4 antagonist displaying an IC50 of 15 nM. It effectively inhibits the cytosolic calcium increase induced by CXCL12, with an IC50 value of 1.3 nM [1].

    价 格：￥电议型 号：T61650产 地：中国大陆

  • T61603H3R antagonist 2；化合物 H3R antagonist 2H3R antagonist 2

    H3R antagonist 2 (Compound 23) is a multitarget histamine H3 receptor antagonist. It exhibits inhibitory effects on acetylcholinesterase, butyrylcholinesterase, and human monoamine oxidase B (hMAO B) with IC50 values of 180 nM, 880 nM, and 775 nM, respectively. With a Ki of 170 nM for hH3R, H3R antagonist 2 demonstrates favorable anti-neuropathic pain and memory-enhancing effects. Additionally, it can cross the blood-brain barrier (BBB) [1].

    价 格：￥电议型 号：T61603产 地：中国大陆

  • T61601TLR7/8 antagonist 2；化合物 TLR7/8 antagonist 2TLR7/8 antagonist 2

    TLR7/8 antagonist 2 (Compound 15) is a highly potent and orally active agonist of TLR7/8, exhibiting IC50 values of 4.9 and 0.6 nM for TLR7 and TLR8, respectively. Its strong affinity for these receptors makes it a promising candidate for the treatment and investigation of autoimmune diseases, including lupus erythematosus, which is associated with inappropriate activation of TLR7 and TLR8. Consequently, TLR7/8 antagonist 2 represents a valuable tool for research in the field of autoimmune disea

    价 格：￥电议型 号：T61601产 地：中国大陆

  • T61566P2X7 receptor antagonist-2；化合物 P2X7 receptor antagonist-2P2X7 receptor antagonist-2

    P2X7 receptor antagonist-2 is a highly potent antagonist of the P2X7 receptor, exhibiting a pIC50 value range of 6.5-7.5. Its efficacy in combating neuroinflammation has been demonstrated [1].

    价 格：￥电议型 号：T61566产 地：中国大陆

  • T61536A1AR antagonist 4；化合物 A1AR antagonist 4A1AR antagonist 4

    A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1].

    价 格：￥电议型 号：T61536产 地：中国大陆

  • T61470NMDA receptor antagonist 5；化合物 NMDA receptor antagonist 5NMDA receptor antagonist 5

    NMDA receptor antagonist 5 (Compound 10e), a potent and non-toxic NMDA receptor antagonist, exhibits brain permeability. It is of significance in studying neurological disorders [1].

    价 格：￥电议型 号：T61470产 地：中国大陆

  • T61447CXCR2 antagonist 4；化合物 CXCR2 antagonist 4CXCR2 antagonist 4

    CXCR2 antagonist 4 (compound 7) is a highly potent antagonist that inhibits CXCR2 with an IC50 value of 0.13 μM. It also effectively inhibits the cytosolic calcium increase induced by CXCL8, with an IC50 value of 27 μM. CXCR2 antagonist 4 shows promising potential for anticancer research [1].

    价 格：￥电议型 号：T61447产 地：中国大陆

  • T61420CXCR4 antagonist 6；化合物 CXCR4 antagonist 6CXCR4 antagonist 6

    CXCR4 antagonist 6 (compound 46) is a highly potent inhibitor of CXCR4 with an IC50 value of 79 nM. It effectively inhibits the cytosolic calcium flux induced by CXCL12, achieving an IC50 of 0.25 nM. Moreover, CXCR4 antagonist 6 demonstrates significant mitigation of cell migration mediated by the CXCL12/CXCR4 interaction. Notably, this compound exhibits remarkable efficacy in a mouse model of cancer metastasis [1].

    价 格：￥电议型 号：T61420产 地：中国大陆

  • T61419CXCR4 antagonist 5；化合物 CXCR4 antagonist 5CXCR4 antagonist 5

    CXCR4 antagonist 5 (compound 23), a potent CXCR4 antagonist, exhibits high inhibition efficacy against CXCR4 with an IC50 value of 8.8 nM. It effectively suppresses CXCL12-induced cytosolic calcium increase (IC50 = 0.02 nM) and hinders CXCR4/CXCL12-mediated chemotaxis. Moreover, Compound 23 demonstrates favorable physicochemical properties and in vitro safety profiles, exhibiting only marginal to moderate inhibition of CYP isozymes and hERG [1].

    价 格：￥电议型 号：T61419产 地：中国大陆

  • T61409CXCR4 antagonist 3；化合物 CXCR4 antagonist 3CXCR4 antagonist 3

    CXCR4 antagonist 3 (compound 12a), an effective antagonist of CXCR4, exhibits an IC50 of 11 nM. It is a congener of TIQ15, showcasing exceptional properties such as CXCR4 antagonism, CYP 2D6 inhibition, metabolic stability, and permeability. With its potential for research on the human immunodeficiency virus, CXCR4 antagonist 3 holds great promise [1].

    价 格：￥电议型 号：T61409产 地：中国大陆

  • T61386CXCR2 antagonist 2；化合物 CXCR2 antagonist 2CXCR2 antagonist 2

    CXCR2 antagonist 2 is a potent CXCR2 antagonist for cancer immunotherapy with an IC 50 value of 95 nM.

    价 格：￥电议型 号：T61386产 地：中国大陆

  • T61363CXCR4 antagonist 8；化合物 CXCR4 antagonist 8CXCR4 antagonist 8

    CXCR4 antagonist 8 (Compound 3) is a potent inhibitor of CXCR4. It demonstrates an IC50 value of 57 nM in CXCR4 antagonism. In addition, it effectively inhibits the increase in cytosolic calcium induced by CXCL12 with an IC50 value of 0.24 nM. Furthermore, Compound 3 shows efficacy in the inhibition of CXCL12/CXCR4-mediated cell migration [1].

    价 格：￥电议型 号：T61363产 地：中国大陆

  • T61359CXCR2 antagonist 6；化合物 CXCR2 antagonist 6CXCR2 antagonist 6

    CXCR2 antagonist 6 (compound 35c) is a potent CXCR2 antagonist. CXCR2 antagonist 6 shows potent CXCR2 binding affinity ( IC 50 =0.044 μM) and calcium mobilization ( IC 50 =0.66 μM) [ 1].

    价 格：￥电议型 号：T61359产 地：中国大陆

  • T61357EP3 antagonist 3；化合物 EP3 antagonist 3EP3 antagonist 3

    EP3 antagonist 3 (compound 2) is a highly effective and specific antagonist of the EP3 receptor. It displays significant oral bioavailability and exhibits a strong pKi value of 8.3. Furthermore, EP3 antagonist 3 possesses excellent pharmacokinetic characteristics, making it a suitable candidate for experimental investigations involving overactive bladder (OAB) research [1].

    价 格：￥电议型 号：T61357产 地：中国大陆

  • T61356CXCR2 antagonist 3；化合物 CXCR2 antagonist 3CXCR2 antagonist 3

    CXCR2 antagonist 3 (compound 11h) is a highly effective antagonist of CXC chemokine receptor 2 (CXCR2). It displays potent activity in inhibiting neutrophil infiltration into the air pouch, with double-digit nanomolar potencies against CXCR2. Moreover, CXCR2 antagonist 3 reduces the infiltration of neutrophils and MDSCs, while enhancing the infiltration of CD3+ T lymphocytes into Pan02 tumor tissues [1].

    价 格：￥电议型 号：T61356产 地：中国大陆

  • T61347D4R antagonist-1；化合物 D4R antagonist-1D4R antagonist-1

    D4R Antagonist-1, characterized by its potent and selective antagonistic action against D4 receptors with an IC50 value of 6.87 μM, holds potential for Parkinson’s disease research [1].

    价 格：￥电议型 号：T61347产 地：中国大陆

  • T61236CXCR2 antagonist 7；化合物 CXCR2 antagonist 7CXCR2 antagonist 7

    CXCR2 antagonist 7 (compound 19) is a potent CXCR2 antagonist. CXCR2 antagonist 7 shows potent CXCR2 binding affinity ( IC 50 =0.044 μM) and calcium mobilization ( IC 50 =0.66 μM) [ 1].

    价 格：￥电议型 号：T61236产 地：中国大陆

  • T61235CXCR2 antagonist 5；化合物 CXCR2 antagonist 5CXCR2 antagonist 5

    CXCR2 antagonist 5 (compound 25) is a potent CXCR2 antagonist. CXCR2 antagonist 5 shows potent CXCR2 binding affinity ( IC 50 =0.013 μM) and calcium mobilization ( IC 50 =0.1 μM) [ 1].

    价 格：￥电议型 号：T61235产 地：中国大陆

  • T61144Hepcidin antagonist-1；Hepcidin 拮抗剂1Hepcidin antagonist-1

    Hepcidin antagonist-1 is an iron-modulating antagonist.Hepcidin antagonist-1 can be used to study metabolic disorders such as iron-deficiency diseases and anemia.

    价 格：￥电议型 号：T61144产 地：中国大陆

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