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T61419CXCR4 antagonist 5；化合物 CXCR4 antagonist 5CXCR4 antagonist 5
CXCR4 antagonist 5 (compound 23), a potent CXCR4 antagonist, exhibits high inhibition efficacy against CXCR4 with an IC50 value of 8.8 nM. It effectively suppresses CXCL12-induced cytosolic calcium increase (IC50 = 0.02 nM) and hinders CXCR4/CXCL12-mediated chemotaxis. Moreover, Compound 23 demonstrates favorable physicochemical properties and in vitro safety profiles, exhibiting only marginal to moderate inhibition of CYP isozymes and hERG [1].
价 格：￥电议型 号：T61419产 地：中国大陆
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T61409CXCR4 antagonist 3；化合物 CXCR4 antagonist 3CXCR4 antagonist 3
CXCR4 antagonist 3 (compound 12a), an effective antagonist of CXCR4, exhibits an IC50 of 11 nM. It is a congener of TIQ15, showcasing exceptional properties such as CXCR4 antagonism, CYP 2D6 inhibition, metabolic stability, and permeability. With its potential for research on the human immunodeficiency virus, CXCR4 antagonist 3 holds great promise [1].
价 格：￥电议型 号：T61409产 地：中国大陆
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T61386CXCR2 antagonist 2；化合物 CXCR2 antagonist 2CXCR2 antagonist 2
CXCR2 antagonist 2 is a potent CXCR2 antagonist for cancer immunotherapy with an IC 50 value of 95 nM.
价 格：￥电议型 号：T61386产 地：中国大陆
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T61363CXCR4 antagonist 8；化合物 CXCR4 antagonist 8CXCR4 antagonist 8
CXCR4 antagonist 8 (Compound 3) is a potent inhibitor of CXCR4. It demonstrates an IC50 value of 57 nM in CXCR4 antagonism. In addition, it effectively inhibits the increase in cytosolic calcium induced by CXCL12 with an IC50 value of 0.24 nM. Furthermore, Compound 3 shows efficacy in the inhibition of CXCL12/CXCR4-mediated cell migration [1].
价 格：￥电议型 号：T61363产 地：中国大陆
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T61359CXCR2 antagonist 6；化合物 CXCR2 antagonist 6CXCR2 antagonist 6
CXCR2 antagonist 6 (compound 35c) is a potent CXCR2 antagonist. CXCR2 antagonist 6 shows potent CXCR2 binding affinity ( IC 50 =0.044 μM) and calcium mobilization ( IC 50 =0.66 μM) [ 1].
价 格：￥电议型 号：T61359产 地：中国大陆
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T61357EP3 antagonist 3；化合物 EP3 antagonist 3EP3 antagonist 3
EP3 antagonist 3 (compound 2) is a highly effective and specific antagonist of the EP3 receptor. It displays significant oral bioavailability and exhibits a strong pKi value of 8.3. Furthermore, EP3 antagonist 3 possesses excellent pharmacokinetic characteristics, making it a suitable candidate for experimental investigations involving overactive bladder (OAB) research [1].
价 格：￥电议型 号：T61357产 地：中国大陆
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T61356CXCR2 antagonist 3；化合物 CXCR2 antagonist 3CXCR2 antagonist 3
CXCR2 antagonist 3 (compound 11h) is a highly effective antagonist of CXC chemokine receptor 2 (CXCR2). It displays potent activity in inhibiting neutrophil infiltration into the air pouch, with double-digit nanomolar potencies against CXCR2. Moreover, CXCR2 antagonist 3 reduces the infiltration of neutrophils and MDSCs, while enhancing the infiltration of CD3+ T lymphocytes into Pan02 tumor tissues [1].
价 格：￥电议型 号：T61356产 地：中国大陆
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T61347D4R antagonist-1；化合物 D4R antagonist-1D4R antagonist-1
D4R Antagonist-1, characterized by its potent and selective antagonistic action against D4 receptors with an IC50 value of 6.87 μM, holds potential for Parkinson’s disease research [1].
价 格：￥电议型 号：T61347产 地：中国大陆
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T61236CXCR2 antagonist 7；化合物 CXCR2 antagonist 7CXCR2 antagonist 7
CXCR2 antagonist 7 (compound 19) is a potent CXCR2 antagonist. CXCR2 antagonist 7 shows potent CXCR2 binding affinity ( IC 50 =0.044 μM) and calcium mobilization ( IC 50 =0.66 μM) [ 1].
价 格：￥电议型 号：T61236产 地：中国大陆
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T61235CXCR2 antagonist 5；化合物 CXCR2 antagonist 5CXCR2 antagonist 5
CXCR2 antagonist 5 (compound 25) is a potent CXCR2 antagonist. CXCR2 antagonist 5 shows potent CXCR2 binding affinity ( IC 50 =0.013 μM) and calcium mobilization ( IC 50 =0.1 μM) [ 1].
价 格：￥电议型 号：T61235产 地：中国大陆
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T61181Pentagamavunon-1；化合物 Pentagamavunon-1Pentagamavunon-1
Pentagamavunon-1 (PGV-1) is an oral Curcumin analog that effectively induces apoptosis through multiple molecular mechanisms. It primarily targets and inhibits key angiogenic factors, including cyclooxygenase-2 (COX-2) and vascular endothelial growth factor (VEGF), which play crucial roles in mediating cell proliferation and survival. Additionally, PGV-1 possesses the ability to inhibit the activation of NF-κB, further enhancing its apoptotic effects. [1]
价 格：￥电议型 号：T61181产 地：中国大陆
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T61144Hepcidin antagonist-1；Hepcidin 拮抗剂1Hepcidin antagonist-1
Hepcidin antagonist-1 is an iron-modulating antagonist.Hepcidin antagonist-1 can be used to study metabolic disorders such as iron-deficiency diseases and anemia.
价 格：￥电议型 号：T61144产 地：中国大陆
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T61068AMPA receptor antagonist-2；AMPA受体拮抗剂2AMPA receptor antagonist-2
AMPA receptor antagonist-2 is an AMPA receptor antagonist.
价 格：￥电议型 号：T61068产 地：中国大陆
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T61064nAChR antagonist 1；化合物 nAChR antagonist 1nAChR antagonist 1
nAChR antagonist 1 (compound B15) is a highly effective antagonist of α7 nAChR, demonstrating an IC50 value of 3.3 μM. Its versatility makes it an ideal candidate for investigating the pathogenesis of schizophrenia, Alzheimer´s disease, and inflammatory disorders [1].
价 格：￥电议型 号：T61064产 地：中国大陆
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T61026CaV1.3 antagonist-1；化合物 CaV1.3 antagonist-1CaV1.3 antagonist-1
CaV1.3 antagonist-1 is a cyclopentyl derivative with the potential for the research of Parkinson´s disease. CaV1.3 antagonist-1 inhibits Ca V 1.3 LTCC over 600-fold more effectively than Ca V 1.2 LTCC. CaV1.3 antagonist-1 is a potent and highly selective antagonist of Ca V 1.3 L-type calcium channel (LTCC) with an IC50 value of 1.7 μM [1].
价 格：￥电议型 号：T61026产 地：中国大陆
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T60988Androgen receptor antagonist 4；化合物 Androgen receptor antagonist 4Androgen receptor antagonist 4
Androgen receptor antagonist 4 (Compound AT2) has anticancer activities. Androgen receptor antagonist 4 potently antagonizes the activity of AR transcriptional, inhibits downstream target gene of AR, and blocks the DHT-induced nuclear translocation of AR. Androgen receptor antagonist 4 is an antagonist of androgen receptor (AR) (IC 50 = 0.15 μM) [1].
价 格：￥电议型 号：T60988产 地：中国大陆
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T60987Androgen receptor antagonist 3；化合物 Androgen receptor antagonist 3Androgen receptor antagonist 3
Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].
价 格：￥电议型 号：T60987产 地：中国大陆
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T60917Dopamine D4 receptor antagonist-1；化合物 Dopamine D4 receptor antagonist-1Dopamine D4 receptor antagoni
Dopamine D4 receptor antagonist-1 can be used in schizophrenia study. Dopamine D4 receptor antagonist-1 is a selective antagonist of Dopamine D4 receptor (DRD4). The Ki value of Dopamine D4 receptor antagonist-1 for Hd4.2 is 9.0 nM [1].
价 格：￥电议型 号：T60917产 地：中国大陆
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T60915A1AR antagonist 5；化合物 A1AR antagonist 5A1AR antagonist 5
A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].
价 格：￥电议型 号：T60915产 地：中国大陆
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T60872Adenosine receptor antagonist 3；化合物 Adenosine receptor antagonist 3Adenosine receptor antagonist 3
Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].
价 格：￥电议型 号：T60872产 地：中国大陆
