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T62054D4R antagonis-2；化合物 D4R antagonis-2D4R antagonis-2
D4R antagonist-2 is a potent and selective D4R antagonist (IC50= 6.52 μM). D4R antagonist-2 displays favorable in vitro PK parameters and exhibits good brain penetration. D4R antagonist-2 has the research potential in Parkinson’s disease.
价 格：￥电议型 号：T62054产 地：中国大陆
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T62050Orexin receptor antagonist 4；化合物 Orexin receptor antagonist 4Orexin receptor antagonist 4
Orexin receptor antagonist 4 is potent and selective orexin 2 receptor (OX2R) antagonist. Orexin receptor antagonist 4 shows IC50 of 4.27 nM and 295 nM for OX2R and OX1R, respectively.
价 格：￥电议型 号：T62050产 地：中国大陆
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T61989CB1R antagonist 1；CB1R拮抗剂1CB1R antagonist 1
CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
价 格：￥电议型 号：T61989产 地：中国大陆
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T61923ERRα antagonist-2；化合物 ERRα antagonist-2ERRα antagonist-2
ERRα antagonist-2 (Compound 11) is a potential Reverse agonist of ERR α (estrogen receptor related receptor α) (IC50=0.80 μ M). ERRα antagonist-2 can inhibit the migration and invasion of ER-negative MDA-MB-231 cells. ERRα antiagonist-2 inhibits the growth of breast cancer in vivo.
价 格：￥电议型 号：T61923产 地：中国大陆
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T61909Estrogen receptor antagonist 7；化合物 Estrogen receptor antagonist 7Estrogen receptor antagonist 7
Estrogen Receptor Antagonist 7 (Compound 13) is a potent antagonist of estrogen receptors (ER), demonstrating antiproliferative effects against breast and ovarian cancer cells, along with anticancer and anti-uterotrophic activities [1].
价 格：￥电议型 号：T61909产 地：中国大陆
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T618375-HT6/5-HT2AR antagonist-1；化合物 5-HT6/5-HT2AR antagonist-15-HT6/5-HT2AR antagonist-1
5-HT6/5-HT2AR antagonist-1 is a powerful and effective compound that acts as a dual antagonist for both the 5-HT6 and 5-HT2A receptors. It exhibits high potency with K i values of 11 nM and 39 nM for the respective receptors [1].
价 格：￥电议型 号：T61837产 地：中国大陆
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T61813AMPA receptor antagonist-3；AMPA受体拮抗剂3AMPA receptor antagonist-3
AMPA receptor antagonist-3 is an AMPA receptor antagonist.
价 格：￥电议型 号：T61813产 地：中国大陆
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T61811GPVI antagonist 3；化合物 GPVI antagonist 3GPVI antagonist 3
GPVI antagonist 3 (Compound 2) is a potential antagonist that shows promising antiplatelet activity by selectively inhibiting the interaction between the Glycoprotein VI (GPVI) receptor and its ligands. It demonstrates potent inhibitory effects, with IC50 values of 1.01 μM for collagen, 1.92 μM for CRP, 7.24 μM for convulxin, and 51.74 μM for thrombin. GPVI is a major collagen receptor on platelets, making it an ideal target for safe and effective antithrombotic treatment. Therefore, GPVI antago
价 格：￥电议型 号：T61811产 地：中国大陆
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T618075-HT6/7 antagonist 1；5-HT6/7拮抗剂15-HT6/7 antagonist 1
5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer´s disease.
价 格：￥电议型 号：T61807产 地：中国大陆
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T61788TRPV1 antagonist 3；化合物 TRPV1 antagonist 3TRPV1 antagonist 3
TRPV1 antagonist 3 (Compound 7q) is a highly potent antagonist of the TRPV1 receptor with an IC50 of 2.66 nM against capsaicin. It exhibits selectivity towards its mode of action and is orally bioavailable (with a bioavailability of 60%). Additionally, it can penetrate the central nervous system [1].
价 格：￥电议型 号：T61788产 地：中国大陆
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T61744A1/A3 AR antagonist 2；化合物 A1/A3 AR antagonist 2A1/A3 AR antagonist 2
The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.
价 格：￥电议型 号：T61744产 地：中国大陆
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T61697GPVI antagonist 1；化合物 GPVI antagonist 1GPVI antagonist 1
GPVI antagonist 1 (compound 5) functions as an antagonist for the glycoprotein VI (GPVI) platelet receptor. It effectively inhibits collagen-induced platelet aggregation, demonstrating an IC50 value of 25.3 μM [1].
价 格：￥电议型 号：T61697产 地：中国大陆
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T61650CXCR4 antagonist 9；化合物 CXCR4 antagonist 9CXCR4 antagonist 9
CXCR4 antagonist 9 (Compound 2) is a potent CXCR4 antagonist displaying an IC50 of 15 nM. It effectively inhibits the cytosolic calcium increase induced by CXCL12, with an IC50 value of 1.3 nM [1].
价 格：￥电议型 号：T61650产 地：中国大陆
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T61603H3R antagonist 2；化合物 H3R antagonist 2H3R antagonist 2
H3R antagonist 2 (Compound 23) is a multitarget histamine H3 receptor antagonist. It exhibits inhibitory effects on acetylcholinesterase, butyrylcholinesterase, and human monoamine oxidase B (hMAO B) with IC50 values of 180 nM, 880 nM, and 775 nM, respectively. With a Ki of 170 nM for hH3R, H3R antagonist 2 demonstrates favorable anti-neuropathic pain and memory-enhancing effects. Additionally, it can cross the blood-brain barrier (BBB) [1].
价 格：￥电议型 号：T61603产 地：中国大陆
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T61601TLR7/8 antagonist 2；化合物 TLR7/8 antagonist 2TLR7/8 antagonist 2
TLR7/8 antagonist 2 (Compound 15) is a highly potent and orally active agonist of TLR7/8, exhibiting IC50 values of 4.9 and 0.6 nM for TLR7 and TLR8, respectively. Its strong affinity for these receptors makes it a promising candidate for the treatment and investigation of autoimmune diseases, including lupus erythematosus, which is associated with inappropriate activation of TLR7 and TLR8. Consequently, TLR7/8 antagonist 2 represents a valuable tool for research in the field of autoimmune disea
价 格：￥电议型 号：T61601产 地：中国大陆
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T61566P2X7 receptor antagonist-2；化合物 P2X7 receptor antagonist-2P2X7 receptor antagonist-2
P2X7 receptor antagonist-2 is a highly potent antagonist of the P2X7 receptor, exhibiting a pIC50 value range of 6.5-7.5. Its efficacy in combating neuroinflammation has been demonstrated [1].
价 格：￥电议型 号：T61566产 地：中国大陆
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T61536A1AR antagonist 4；化合物 A1AR antagonist 4A1AR antagonist 4
A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1].
价 格：￥电议型 号：T61536产 地：中国大陆
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T61470NMDA receptor antagonist 5；化合物 NMDA receptor antagonist 5NMDA receptor antagonist 5
NMDA receptor antagonist 5 (Compound 10e), a potent and non-toxic NMDA receptor antagonist, exhibits brain permeability. It is of significance in studying neurological disorders [1].
价 格：￥电议型 号：T61470产 地：中国大陆
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T61447CXCR2 antagonist 4；化合物 CXCR2 antagonist 4CXCR2 antagonist 4
CXCR2 antagonist 4 (compound 7) is a highly potent antagonist that inhibits CXCR2 with an IC50 value of 0.13 μM. It also effectively inhibits the cytosolic calcium increase induced by CXCL8, with an IC50 value of 27 μM. CXCR2 antagonist 4 shows promising potential for anticancer research [1].
价 格：￥电议型 号：T61447产 地：中国大陆
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T61420CXCR4 antagonist 6；化合物 CXCR4 antagonist 6CXCR4 antagonist 6
CXCR4 antagonist 6 (compound 46) is a highly potent inhibitor of CXCR4 with an IC50 value of 79 nM. It effectively inhibits the cytosolic calcium flux induced by CXCL12, achieving an IC50 of 0.25 nM. Moreover, CXCR4 antagonist 6 demonstrates significant mitigation of cell migration mediated by the CXCL12/CXCR4 interaction. Notably, this compound exhibits remarkable efficacy in a mouse model of cancer metastasis [1].
价 格：￥电议型 号：T61420产 地：中国大陆
