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T73004METTL3-IN-3；化合物 METTL3-IN-3METTL3-IN-3
METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor [1] .
价 格：￥电议型 号：T73004产 地：中国大陆
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T72989hGGPPS-IN-3；化合物 hGGPPS-IN-3hGGPPS-IN-3
Compound 13h (hGGPPS-IN-3) is a potent inhibitor of human geranylgeranyl pyrophosphate synthase (hGGPPS), characterized as a C-2-substituted thienopyrimidine-based bisphosphonate analogue (C2-ThP-BPs). It selectively induces apoptosis in multiple myeloma (MM) cells and demonstrates antimyeloma activity in vivo [1].
价 格：￥电议型 号：T72989产 地：中国大陆
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T72933ChemR23-IN-3；化合物 ChemR23-IN-3ChemR23-IN-3
ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.
价 格：￥电议型 号：T72933产 地：中国大陆
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T72890VEGFR-2-IN-30；化合物 VEGFR-2-IN-30VEGFR-2-IN-30
VEGFR-2-IN-30, a compound acting primarily as a VEGFR-2 inhibitor (IC50: 66 nM), demonstrates additional inhibitory effects on PDGFR, EGFR, and FGFR1, with IC50 values of 180, 98, and 82 nM, respectively. It effectively arrests cancer cells in the S-phase and induces both early and late apoptosis.
价 格：￥电议型 号：T72890产 地：中国大陆
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T72875sEH/AChE-IN-3；化合物 sEH/AChE-IN-3sEH/AChE-IN-3
sEH/AChE-IN-3 (15) serves as a dual inhibitor targeting both soluble epoxide hydrolase (sEH) and acetylcholinesterase (AChE), demonstrating potent activity and the ability to cross the blood-brain barrier (BBB). It exhibits IC50 values of 0.4 nM for human sEH (hsEH), 1.94 nM for human AChE (hAChE), 615 nM for human butyrylcholinesterase (hBChE), 4.3 nM for mouse sEH (msEH), and 2.61 nM for mouse AChE (mAChE), indicating its efficacy across these enzymes.
价 格：￥电议型 号：T72875产 地：中国大陆
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T72791AChE/MAO-B-IN-3；化合物 AChE/MAO-B-IN-3AChE/MAO-B-IN-3
AChE/MAO-B-IN-3 is a dual inhibitor targeting both acetylcholinesterase (AChE) and monoamine oxidase B (MAO-B), exhibiting inhibitory concentrations (IC50s) of 0.0257 μM and 0.0456 μM against human AChE and MAO-B, respectively. This compound holds potential for Alzheimer’s disease research.
价 格：￥电议型 号：T72791产 地：中国大陆
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T72777c-Met/HDAC-IN-3；化合物 c-Met/HDAC-IN-3c-Met/HDAC-IN-3
c-Met/HDAC-IN-3, a dual inhibitor targeting both c-Met and HDAC, exhibits potent inhibitory activity with IC50 values of 12.50 nM for c-Met and 26.97 nM for HDAC1. It induces apoptosis and causes cell cycle arrest in the G2/M phase.
价 格：￥电议型 号：T72777产 地：中国大陆
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T72724PD-1/PD-L1-IN-30；化合物 PD-1/PD-L1-IN-30PD-1/PD-L1-IN-30
PD-1/PD-L1-IN-30 is a PD-1/PD-L1 binding inhibitor, with an IC 50 value of 0.018 μM. PD-1/PD-L1-IN-30 can be used for research of cancers and other related diseases [1] .
价 格：￥电议型 号：T72724产 地：中国大陆
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T72718SARS-CoV-2-IN-36；化合物 SARS-CoV-2-IN-36SARS-CoV-2-IN-36
SARS-CoV-2-IN-36 is a potent inhibitor of SARS-CoV-2 Mpro (SARS-CoV), demonstrating an IC50 of 2.37 μM and a Kd of 1.19 μM in enzymatic assays. This compound exhibits antiviral activity against SARS-CoV-2 variants UC-1074, RG2674, and NVDBB-2220 in Vero cells.
价 格：￥电议型 号：T72718产 地：中国大陆
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T72701Cavα2δ1&NET-IN-3；化合物 Cavα2δ1&NET-IN-3Cavα2δ1&NET-IN-3
Cavα2δ1&NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET). It exhibits inhibitory constants (Ki) ranging from 100 to 500 nM for the human α2δ-1 subunit of the Ca v 2.2 calcium channel and NET, respectively.
价 格：￥电议型 号：T72701产 地：中国大陆
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T72504Aurora Kinases-IN-3；化合物 Aurora Kinases-IN-3Aurora Kinases-IN-3
Aurora Kinases-IN-3, an orally active inhibitor of AURKB, suppresses AURKB activity by hindering its mitotic localization rather than by inhibiting its phosphorylation of H3 at Ser10.
价 格：￥电议型 号：T72504产 地：中国大陆
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T72453AChE/BChE/MAO-B-IN-3；化合物 AChE/BChE/MAO-B-IN-3AChE/BChE/MAO-B-IN-3
AChE/BChE/MAO-B-IN-3, an indan-1-one derivative, serves as a potent inhibitor of human monoamine oxidase B (MAO-B) with an IC50 of 0.0359 μM, demonstrating significant inhibitory effects on acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) with IC50 values of 0.0473 μM and 0.0782 μM, respectively. Exhibiting notable antioxidant activity, AChE/BChE/MAO-B-IN-3 holds considerable promise for Alzheimer´s disease (AD) research.
价 格：￥电议型 号：T72453产 地：中国大陆
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T72372Neuroinflammatory-IN-3；化合物 Neuroinflammatory-IN-3Neuroinflammatory-IN-3
Neuroinflammatory-IN-3 is a tubulin inhibitor that serves as both an anti-neuroinflammatory agent and a potent antitumor agent by inhibiting tubulin polymerization.
价 格：￥电议型 号：T72372产 地：中国大陆
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T72299Mtb-cyt-bd oxidase-IN-3；化合物 Mtb-cyt-bd oxidase-IN-3Mtb-cyt-bd oxidase-IN-3
Mtb-cyt-bd oxidase-IN-3, an inhibitor of Mycobacterium tuberculosis cytochrome bd oxidase (Mtb cyt-bd oxidase), exhibits an IC50 value of 0.36 μM and demonstrates an ability to inhibit the growth of Mycobacterium tuberculosis with an MIC of 32 μM. This compound is utilized in tuberculosis research.
价 格：￥电议型 号：T72299产 地：中国大陆
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T72203Reverse transcriptase-IN-3；化合物 Reverse transcriptase-IN-3Reverse transcriptase-IN-3
Reverse transcriptase-IN-3, a pyrimidine-5-carboxamide derivative, functions as an inhibitor of HIV-1, demonstrating potent activity against both wild-type and mutant strains of HIV-1.
价 格：￥电议型 号：T72203产 地：中国大陆
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T72167Tubulin polymerization-IN-39；化合物 Tubulin polymerization-IN-39Tubulin polymerization-IN-39
Tubulin polymerization-IN-39, a tubulin polymerization inhibitor with an IC50 of 4.9 μM, targets the colchicine-binding site to hinder tubulin polymerization. This compound effectively suppresses cancer cell proliferation.
价 格：￥电议型 号：T72167产 地：中国大陆
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T72165Xanthine oxidoreductase-IN-3；黄氨酸氧化还原酶抑制剂3Xanthine oxidoreductase-IN-3
Xanthine oxidoreductase-IN-3 is an orally active xanthine oxidoreductase (XOR) inhibitor (IC50: 26.3 nM).Xanthine oxidoreductase-IN-3 can be used in acute hyperuricemia studies.
价 格：￥电议型 号：T72165产 地：中国大陆
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T72137Mitochondrial respiration-IN-3；化合物 Mitochondrial respiration-IN-3Mitochondrial respiration-IN-3
Mitochondrial respiration-IN-3, a fluorine derivative of Dalfopristin, possesses cell membrane permeability and exhibits the capability to inhibit mitochondrial translation in glioblastoma stem cells. This compound is utilized in cancer research [1].
价 格：￥电议型 号：T72137产 地：中国大陆
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T72109Werner syndrome RecQ helicase-IN-3；化合物 Werner syndrome RecQ helicase-IN-3Werner syndrome RecQ helica
Werner syndrome RecQ helicase-IN-3, a potent and orally active inhibitor of Werner syndrome RecQ helicase (WRN), exhibits anticancer and antiproliferative activities with an IC50 value of 0.06 ?M.
价 格：￥电议型 号：T72109产 地：中国大陆
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T72098Eleven-Nineteen-Leukemia Protein IN-3；化合物 Eleven-Nineteen-Leukemia Protein IN-3Eleven-Nineteen-Leuke
Eleven-Nineteen-Leukemia Protein IN-3, an orally active ENL YEATS domain inhibitor, exhibits potent activity with an IC50 of 15.4 nM. It downregulates MYC expression via ENL in cells and enhances ENL protein´s thermal stability in vitro [1].
价 格：￥电议型 号：T72098产 地：中国大陆
