T6117TivantinibARQ 197

Tivantinib is an orally bioavailable small molecule inhibitor of c-Met with potential antineoplastic activity.

价 格：￥电议型 号：T6117产 地：中国大陆

T6116Bleomycin Sulfate硫酸博来霉素；硫酸博莱霉素；Blenoxane；NSC125066

Bleomycin Sulfate, a glycopeptide antibiotic, is an anticancer agent for squamous cell carcinomas (SCC). In UT-SCC-19A cells, the IC50 of Bleomycin Sulfate is 4 nM.

价 格：￥电议型 号：T6116产 地：中国大陆

T6115Fostamatinib福他替尼；R788

Fostamatinib(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.

价 格：￥电议型 号：T6115产 地：中国大陆

T6114Nifursol硝呋索尔；尼呋索尔

Nifursol is a livestock feed additive and antiobiotic used to prevent the growth of histomonas.

价 格：￥电议型 号：T6114产 地：中国大陆

T6113ICG-001

ICG-001 antagonizes Wnt/β-catenin/TCF-mediated transcription and specifically binds to element-binding protein (CBP) with IC50 of 3 μM, but is not the related transcriptional coactivator p300.

价 格：￥电议型 号：T6113产 地：中国大陆

T6112Doxercalciferol度骨化醇；1.alpha.-Hydroxyvitamin D2；1α-hydroxyvitamin D2；Hectorol；TSA 840

Doxercalciferol is a synthetic vitamin D2 analog, suppressing parathyroid synthesis and secretion, used to treat secondary hyperparathyroidism and metabolic bone disease.

价 格：￥电议型 号：T6112产 地：中国大陆

T6111Selisistat司来司他；EX-527；SEN0014196

EX 527 is an effective and specific SIRT1 inhibitor (IC50: 38 nM) and shows >200-fold selectivity against SIRT2/3.

价 格：￥电议型 号：T6111产 地：中国大陆

T6110YM-201636YM201636

YM201636 (IC50=33 nM), a specific PIKfyve inhibitor, is less effective to p110α and insensitive to Fabl, which is yeast orthologue.

价 格：￥电议型 号：T6110产 地：中国大陆

T4611EN300-203561

价 格：￥电议型 号：T4611产 地：中国大陆

T3621BrigatinibAP-26113；布格替尼

Brigatinib is a highly potent and selective ALK inhibitor.

价 格：￥电议型 号：T3621产 地：中国大陆

T3611Sodium Glucuronic Acid葡醛酸钠；4-FLUOROCINNAMONITRILE；Sodium Glucoronic

Sodium Glucuronic Acid is used in the treatment of hepatitis and liver cirrhosis.

价 格：￥电议型 号：T3611产 地：中国大陆

T2611CCT 137690CCT137690

CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).

价 格：￥电议型 号：T2611产 地：中国大陆

T2216EntacaponeOR-611；恩他卡朋

Entacapone is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).

价 格：￥电议型 号：T2216产 地：中国大陆

T21611LBWX 46 AcetateBWX 46 Acetate(172997-92-1 Free base)

BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.

价 格：￥电议型 号：T21611L产 地：中国大陆

T2020RGW 611

Detail unknown.

价 格：￥电议型 号：T2020产 地：中国大陆

T1971WAY-262611WAY262611；WAY 262611

WAY-262611 is a wingless β-Catenin agonist.

价 格：￥电议型 号：T1971产 地：中国大陆

T16118MLS0315771

MLS0315771 is an effective and biologically active competitive phosphomannose isomerase (MPI) inhibitor (IC50: ~1 μM and a Ki: 1.4 μM).

价 格：￥电议型 号：T16118产 地：中国大陆

T16116MLN-4760

MLN-4760 is an angiotensin-converting (ACE2) inhibitor(human ACE2;IC50=0.44 nM). It also has excellent selectivity (>5000-fold) versus related enzymes including human testicular ACE (IC50, >100 μM) and bovine carboxypeptidase A (CPDA; IC50, 27 μM).

价 格：￥电议型 号：T16116产 地：中国大陆

T16115MLi-2

MLi-2 is a structurally novel, highly potent, and selective LRRK2 kinase inhibitor with central nervous system activity. MLi-2 exhibits exceptional potency in a purified LRRK2 kinase assay in vitro (IC50 = 0.76 nM), a cellular assay monitoring dephosphory

价 格：￥电议型 号：T16115产 地：中国大陆

T16110ML418

ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.

价 格：￥电议型 号：T16110产 地：中国大陆