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T70257Avitriptan HCl；化合物 Avitriptan HClAvitriptan HCl
Avitriptan, also known as BMS-180048, is a selective 5-HT1-like receptor agonist. Avitriptan is an effective compound for the treatment of migraine headaches with a prolonged duration of response. Avitriptan Is a Ligand and Agonist of Human Aryl Hydrocarbon Receptor That Induces CYP1A1 in Hepatic and Intestinal Cells.
价 格：￥电议型 号：T70257产 地：中国大陆
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T70233Efegatran HCl；化合物 Efegatran HClEfegatran HCl
Efegatran, also known as GYKI-14166, RGH-2958 and LY294468, a thrombin inhibitor which is being developed by IVAX for the potential treatment of thromboembolic disorders.
价 格：￥电议型 号：T70233产 地：中国大陆
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T70231Osanetant HCl；化合物 Osanetant HClOsanetant HCl
Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonist
价 格：￥电议型 号：T70231产 地：中国大陆
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T70202DDR1-IN-1 dihydrochloride；化合物 DDR1-IN-1 HClDDR1-IN-1 dihydrochloride
DDR1-IN-1 dihydrochloride is a selective and potent inhibitor of the DDR1 receptor tyrosine kinase, exhibiting an IC50 of 105 nM. It demonstrates fourfold reduced potency against DDR2, with an IC50 of 413 nM.
价 格：￥电议型 号：T70202产 地：中国大陆
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T70200VU590 HCl；化合物 VU590 HClVU590 HCl
VU590 is a small molecule inhibitor of KCNJ1 (IC50 = 294 nM).
价 格：￥电议型 号：T70200产 地：中国大陆
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T70199Enecadin HCl；化合物 Enecadin HClEnecadin HCl
Enecadin HCl is a voltage-dependent sodium and calcium channel blocker.
价 格：￥电议型 号：T70199产 地：中国大陆
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T70196AZD1446 HCl；化合物 AZD1446 HClAZD1446 HCl
AZD1446 HCl, also known as TC-6683, is a novel highly selective α4β2 nicotinic acetylcholine receptor agonist for the treatment of cognitive disorders. AZD1446 HCl showed favorable pharmaceutical properties and in vivo efficacy in animal models has been identified as a potential treatment for cognitive deficits associated with psychiatric or neurological conditions and had been evaluated in phase 2 clinical trials as a treatment for Alzheimer´s disease.
价 格：￥电议型 号：T70196产 地：中国大陆
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T70193APC-366 HCl；化合物 APC-366 HClAPC-366 HCl
APC-366 is a selective inhibitor of the mast cell tryptase that inhibits tryptase-induced histamine release from human tonsil and lung cells.
价 格：￥电议型 号：T70193产 地：中国大陆
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T70190Tinostamustine HCl；化合物 Tinostamustine HClTinostamustine HCl
Tinostamustine, also known as EDO-S101, is an alkylatlng histone-deacetylase inhibitor (HDACi) fusion molecule. EDO-S101 is a functional pan-histone-deacetylase inhibitor and is assumed to potentiate the alkylating activity of the compound and/or may help to overcome resistance to other therapeutic agents.
价 格：￥电议型 号：T70190产 地：中国大陆
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T70174Pirlindole-d4 HCl；化合物 Pirlindole-d4 HClPirlindole-d4 HCl
Pirlindole-d4 is intended for use as an internal standard for the quantification of pirlindole by GC- or LC-MS. Pirlindole is a selective and reversible monoamine oxidase A (MAO-A) inhibitor. It is selective for MAO-A over MAO-B. In rats, it reverses the depressive-like effects induced by chronic mild stress (CMS), increases proliferation of hippocampal neural progenitor cells, and reverses dendritic atrophy in granule neurons. Pirlindole is also an inhibitor of enterovirus-D68 and coxsackieviru
价 格：￥电议型 号：T70174产 地：中国大陆
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T70168Tofacitinib HCl；化合物 Tofacitinib HClTofacitinib HCl
Tofacitinib HCl, also known as tasocitinib, CP-690550, is a Janus kinase (JAK) inhibitor. Tofacitinib HCl modulates the signaling pathway at the point of JAKs, preventing the phosphorylation and activation of STATs. JAK enzymes transmit cytokine signaling through pairing of JAKs (e.g., JAK1/JAK3, JAK1/JAK2, JAK1/TyK2, JAK2/JAK2). Tofacitinib HCl inhibited the in vitro activities of JAK1/JAK2, JAK1/JAK3, and JAK2/JAK2 combinations with IC50 of 406, 56, and 1377 nM, respectively.
价 格：￥电议型 号：T70168产 地：中国大陆
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T70164LASSBio-1829 HCl；化合物 LASSBio-1829 HClLASSBio-1829 HCl
LASSBio-1829 HCl is an orally active IKK2 inhibitor.
价 格：￥电议型 号：T70164产 地：中国大陆
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T70161Berotralstat HCl；化合物 Berotralstat HClBerotralstat HCl
Berotralstat HCl is a novel selective inhibitor of plasma kallikrein, blocking the enzymatic activity of plasma kallikrein in releasing bradykinin, the major biologic peptide that promotes swelling and pain associated with attacks of HAE.
价 格：￥电议型 号：T70161产 地：中国大陆
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T70124Tomivosertib HCl；化合物 Tomivosertib HClTomivosertib HCl
Tomivosertib, also known as eFT508 is a MNK1/2 inhibitor. Tomivosertib binds to and inhibits the activity of MNK1 and 2. This prevents MNK1/2-mediated signaling, and inhibits the phosphorylation of certain regulatory proteins, including eukaryotic translation initiation factor 4E (eIF4E), that regulate the translation of messenger RNAs (mRNAs) involved in tumor cell proliferation, angiogenesis, survival and immune signaling.
价 格：￥电议型 号：T70124产 地：中国大陆
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T70096AEG40730 HCl；化合物 AEG40730 HClAEG40730 HCl
AEG40730 is a potent and selective IAP antagonist and a BIR-binding tetrapeptide. AEG40730 binds to cIAP1 and cIAP2, facilitates their autoubiquitination and proteosomal degradation, and causes a dramatic reduction in RIP1 ubiquitination. Treatment with nanomolar concentrations of AEG40730 resulted in the loss of both XIAP and c-IAP1 proteins, albeit with different kinetics.
价 格：￥电议型 号：T70096产 地：中国大陆
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T70077Fadolmidine HCl；化合物 Fadolmidine HClFadolmidine HCl
Fadolmidine, also known as MPV-2426, is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia. Fadolmidine displayed high affinity and full agonist efficacy at all three human alpha2-adrenoceptor subtypes (A, B and C) in transfected CHO cells with EC50 values (nM) of 0.4, 4.9 and 0.5, respectively. Fadolmidine inhibited also electrically evoked contractions in rat vas deferens demonstrating the activation of rodent presynaptic alpha2D-adrenoceptors with an
价 格：￥电议型 号：T70077产 地：中国大陆
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T70063GYKI 52466 HCl；化合物 GYKI 52466 HClGYKI 52466 HCl
GYKI 52466 is an allosteric AMPA receptor antagonist. It selectively inhibits AMPA-induced inward currents (IC50 = 7.5 ?M) over NMDA- or GABA-induced inward currents in primary rat hippocampal neurons at 50 ?M but also inhibits kainate-induced inward currents in the same cells (IC50 = 11 ?M).2 GYKI 52466 (10 ?M) reduces the amplitude of spontaneous excitatory postsynaptic currents (EPSCs) in the same cells. It increases the latency to seizure onset and reduces mortality in a rat model of general
价 格：￥电议型 号：T70063产 地：中国大陆
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T7005LUlixertinib hydrochloride化合物 T7005LUlixertinib HCl|||BVD-523|||VRT752271|||BVD 523|||BVD523|||VRT 75
Ulixertinib is an inhibitor of ERK protein kinase. Downmodulation of ERK protein kinase activity inhibits VEGF secretion by human myeloma cells and myeloma-induced angiogenesis. Upon oral administration, BVD-523 inhibits both ERK 1 and 2, thereby preventing the activation of ERK-mediated signal transduction pathways. This results in the inhibition of ERK-dependent tumor cell proliferation and survival.
价 格：￥电议型 号：T7005L产 地：中国大陆
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T70059ALT-946 HCl；化合物 ALT-946 HClALT-946 HCl
ALT-946 HCl is an inhibitor of advanced glycation that has been shown to improve severe nephropathy in the diabetic transgenic (mREN-2)27 rat.
价 格：￥电议型 号：T70059产 地：中国大陆
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T70044LSarizotan 2HCl；Sarizotan 2盐酸盐Sarizotan 2HCl
Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.
价 格：￥电议型 号：T70044L产 地：中国大陆
