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T15543IA-Alkyne；化合物IA-AlkyneN-Hex-5-ynyl-2-iodo-acetamide|||Iodoacetamide-alkyne；N-Hex-5-ynyl-2-iodo-aceta
IA-Alkyne (Iodoacetamide-alkyne) is a TRP channel (TRPC) agonist. IA-Alkyne can be used to develop an isotopically tagged probe for quantitative cysteine-reactivity profiling. It also has the potential for the study of respiratory infection.
价 格：￥电议型 号：T15543产 地：中国大陆
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T15454GW843682X；化合物GW843682XGW843682；GW843682
GW843682X (GW843682) is a selective and ATP-competitive inhibitor of PLK1 and PLK3 (IC50s = 2.2 nM and 9.1 nM).
价 格：￥电议型 号：T15454产 地：中国大陆
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T15450GW-803430；化合物 T15450GW-3430；GW-3430
GW-803430 is a potent and selective antagonist of melanin-concentrating hormone receptor 1 (MCH R1) (pIC50: 9.3). GW-803430 is orally active in an animal model of obesity.
价 格：￥电议型 号：T15450产 地：中国大陆
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T15443GSK8814；化合物 T15443GSK8814
GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan). GSK8814 displays 500-fold selectivity for ATAD2 over BRD4 BD1. GSK8814 binds to ATAD2 and BRD4 BD1 (pIC50s: 7.3 and 4.6).
价 格：￥电议型 号：T15443产 地：中国大陆
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T15439GSK3395879；化合物 T15439GSK3395879
GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).
价 格：￥电议型 号：T15439产 地：中国大陆
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T15438GSK3186899；化合物GSK31868993,3,3-trifluoro-N-[4-[[3-[(2R)-2-methylmorpholin-4-yl]-1H-pyrazolo[3,4-d]pyr
GSK3186899 is an inhibitor of Cdc2-related kinase 12 with an EC50 of 1.4 μM for L. donovani.
价 格：￥电议型 号：T15438产 地：中国大陆
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T15437GSK3145095；化合物GSK3145095GSK3145095
GSK3145095 is an orally active inhibitor of RIPK1 with IC50 of 5 nM, with potential immunomodulatory activities and antineoplastic.
价 格：￥电议型 号：T15437产 地：中国大陆
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T15436GSK2838232；化合物GSK2838232GSK2838232
GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.
价 格：￥电议型 号：T15436产 地：中国大陆
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T15435GSK2837808A；化合物GSK2837808AGSK2837808A
GSK2837808A is a potent and selective inhibitor of lactate dehydrogenase A (LDHA) (IC50s: 1.9 and 14 nM for LDHA and LDHB, respectively).
价 格：￥电议型 号：T15435产 地：中国大陆
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T15434GSK2798745；化合物 T15434GSK2798745
GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4). It is used in research for the treatment of pulmonary edema associated with congestive heart failure.
价 格：￥电议型 号：T15434产 地：中国大陆
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T15433GSK2795039；化合物GSK2795039GSK2795039
GSK2795039 inhibits reactive oxygen species (ROS) production and NADPH consumption. GSK2795039 decreases apoptosis. GSK2795039 is an inhibitor of NADPH oxidase 2 (NOX2) (pIC50: 6 in different cell-free assays).
价 格：￥电议型 号：T15433产 地：中国大陆
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T15432GSK256073；化合物GSK256073GSK256073
GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 (hydroxy-carboxylic acid receptor 2) full agonist (pEC50: 7.5). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis.
价 格：￥电议型 号：T15432产 地：中国大陆
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T15431Nemiralisib；奈米利塞GSK2269557 (free base)|||GSK2269557；GSK2269557 (free base)|||GSK2269557
Nemiralisib（GSK-2269557 free base） is an orally available, potent and specific PI3Kδ inhibitor with a pKi of 9.9.Nemiralisib is used for the treatment of respiratory diseases including chronic obstructive pulmonary disease.
价 格：￥电议型 号：T15431产 地：中国大陆
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T15430GSK2256294A；化合物GSK2256294AGSK 2256294；GSK 2256294
GSK2256294A (GSK 2256294) is potent, selective inhibitor of recombinant human, rat and mouse sEH with IC50 of 27 pM, 61 pM and 189 pM, respectively.
价 格：￥电议型 号：T15430产 地：中国大陆
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T1543Naftifine hydrochloride；盐酸萘替芬Naftifungin|||Naftifine HCl|||Naftin|||Exoderil；Naftifungin|||盐酸萘替芬|||N
Naftifine Hydrochloride is the hydrochloride salt form of naftifine, an allylamine derivate with synthetic broad-spectrum antifungal activity. Although the exact mechanism through which naftifine hydrochloride exerts its effect is unknown, it appears to selectively inhibit the enzyme squalene 2, 3-epoxidase, thereby inhibiting the biosynthesis of sterol. This results in a decreased amount of sterols, especially ergosterol which is the primary fungal membrane sterol, and a corresponding accumulat
价 格：￥电议型 号：T1543产 地：中国大陆
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T15343Fosteabine；阿糖胞苷烷磷酯YNK 01|||Cytarabine ocfosfate；YNK 01|||Cytarabine ocfosfate|||阿糖胞苷烷磷酯
Fosteabine is an oral and prodrug analog of cytarabine. It is resistant to deoxycytidine deaminase.
价 格：￥电议型 号：T15343产 地：中国大陆
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T15286Flindokalner；化合物FlindokalnerBMS-204352；BMS-204352
Flindokalner (BMS-204352) is a potassium channel modulator and a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is a large conductance calcium-activated K channel (BKca) positive modulator. Flindokalner displays a negative modulatory activity at Kv7.1 channels (Ki=3.7 μM) and acts as a negative modulator of GABAA receptors and it also shows anxiolytic efficacy in vivo.
价 格：￥电议型 号：T15286产 地：中国大陆
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T15243Ertiprotafib；化合物 T15243PTP 112；PTP 112
Ertiprotafib is a PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist inhibitor ( IC50s: 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ).
价 格：￥电议型 号：T15243产 地：中国大陆
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T15240Tazemetostat trihydrochloride；化合物 T15240EPZ-6438 trihydrochloride|||E-7438 trihydrochloride；EPZ-6438
Tazemetostat trihydrochloride is a selective and orally available inhibitor of EZH2 (IC50: 4 nM for rat EZH2). It inhibits the activity of human PRC2-containing wild-type EZH2 (Ki: 2.5 nM). It inhibits EZH2 (IC50s: 11 and 16 nM in peptide assay and nucleosome assay).
价 格：￥电议型 号：T15240产 地：中国大陆
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T15169DS-437；化合物 T15169DS-437
DS-437 is a dual PRMT5/7 inhibitor (IC50s: 6 μM). DS-437 also inhibits DNMT3A and DNMT3B (IC50s: 52 and 62 μM). DS-437 inhibits the methylation of FOXP3.
价 格：￥电议型 号：T15169产 地：中国大陆
