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T73255Akt1-IN-1；化合物 Akt1-IN-1Akt1-IN-1
Akt1-IN-1 is a potent and selective inhibitor of Akt1, demonstrating an IC50 of 18.79 nM in MIA PaCa-2 cells, indicating its high efficacy in inhibiting this specific kinase. Notably, it shows no significant teratogenicity, hepatotoxicity, or cardiotoxicity (No Observed Adverse Effect Level > 100 ?M), making it a viable candidate for anticancer research.
价 格：￥电议型 号：T73255产 地：中国大陆
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T73250JAK-IN-17；化合物 JAK-IN-17JAK-IN-17
JAK-IN-17 is a potent inhibitor of JAK . JAK-IN-17 is useful for the research of multiple diseases, particularly ocular, skin, and respiratory diseases.
价 格：￥电议型 号：T73250产 地：中国大陆
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T73249HBV-IN-15；化合物 HBV-IN-15HBV-IN-15
HBV-IN-15, a flavone derivative, acts as a potent inhibitor of covalently closed circular DNA (cccDNA), which is crucial for viral RNA transcription and subsequent viral DNA production. This compound shows promise for research in Hepatitis B Virus (HBV) infection.
价 格：￥电议型 号：T73249产 地：中国大陆
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T73248RET-IN-13；化合物 RET-IN-13RET-IN-13
RET-IN-13, a quinoline-based compound, effectively inhibits the RET kinase, demonstrating IC50 values of 0.5 nM for RET (WT) and 0.9 nM for RET (V804M). It holds promise for research into tumors and intestinal diseases associated with abnormal RET activation.
价 格：￥电议型 号：T73248产 地：中国大陆
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T73242NSD3-IN-1；化合物 NSD3-IN-1NSD3-IN-1
NSD3-IN-1, a histone methyltransferase NSD3 inhibitor, demonstrates an IC50 of 28.58 μM.
价 格：￥电议型 号：T73242产 地：中国大陆
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T73230UT-B-IN-1；化合物 UT-B-IN-1UT-B-IN-1
UT-B-IN-1 (UTBINH-14) is a reversible, competitive, and selective inhibitor of the urea transporter-B (UT-B), demonstrating IC50 values of 10 nM and 25 nM for human and mouse UT-B, respectively. It exhibits low toxicity and superior selectivity against UT-B compared to UT-A isoforms. This compound enhances urine production and decreases urine concentration in mice, making UT-B-IN-1 suitable for research on diuretic mechanisms.
价 格：￥电议型 号：T73230产 地：中国大陆
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T73224AMPK-IN-1；化合物 AMPK-IN-1AMPK-IN-1
AMPK-IN-1 is an activator of the AMP-activated protein kinase (AMPK) enzyme, specifically targeting the α2β2γ1 isoform with an EC50 of 551 nM. It induces phosphorylation of eEF2 independent of the mTORC1 pathway.
价 格：￥电议型 号：T73224产 地：中国大陆
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T73221CASK-IN-1；化合物 CASK-IN-1CASK-IN-1
CASK-IN-1 is a highly potent and selective CASK inhibitor with a K d value of 0.022 μM.
价 格：￥电议型 号：T73221产 地：中国大陆
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T73212Notum-IN-1；化合物 Notum-IN-1Notum-IN-1
Notum-IN-1 is an orally administered, selective, and brain-penetrating compound that acts as an inhibitor of Notum. It effectively inhibits Wnt signaling in vivo in mice.
价 格：￥电议型 号：T73212产 地：中国大陆
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T73202BChE-IN-11；化合物 BChE-IN-11BChE-IN-11
BChE-IN-11, a selective and non-competitive inhibitor of butyrylcholinesterase (BChE), demonstrates potent activity with an inhibitory concentration (IC50) of 2.1 μM. This compound is applicable in Alzheimer´s disease (AD) research.
价 格：￥电议型 号：T73202产 地：中国大陆
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T73194DOCK2-IN-1；化合物 DOCK2-IN-1DOCK2-IN-1
DOCK2-IN-1, an analogue of CPYPP, effectively inhibits DOCK2 (IC50 = 19.1 μM) by reversibly binding to its DHR-2 domain, thereby hindering its catalytic function. This compound obstructs the activation of Rac in lymphocytes, triggered either by chemokine or antigen receptors. Consequently, DOCK2-IN-1 markedly reduces chemotactic responses and T cell activation [1].
价 格：￥电议型 号：T73194产 地：中国大陆
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T73184BChE-IN-15；化合物 BChE-IN-15BChE-IN-15
BChE-IN-15 is a compound characterized as a pseudo-irreversible, covalent inhibitor of butyrylcholinesterase (BChE), demonstrating potent activity with an inhibitory concentration (IC50) of 1.76 nM against human BChE (hBChE).
价 格：￥电议型 号：T73184产 地：中国大陆
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T73175MMP-1-IN-1；化合物 MMP-1-IN-1MMP-1-IN-1
MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM [1] .
价 格：￥电议型 号：T73175产 地：中国大陆
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T73172FOXM1-IN-1；化合物 FOXM1-IN-1FOXM1-IN-1
FOXM1-IN-1 is a potent FOXM1 inhibitor with an IC 50 value of 2.65 ?M. FOXM1-IN-1 shows antiproliferative activity. FOXM1-IN-1 decreases the the expression of FOXM1, PLK1 , CDC25B protein [1] .
价 格：￥电议型 号：T73172产 地：中国大陆
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T73164SOS1-IN-15；SOS1 抑制剂15SOS1-IN-15
SOS1-IN-15 is an orally active and potent SOS1 inhibitor with potential antitumor activity.SOS1-IN-15 is used in the study of colon cancer.
价 格：￥电议型 号：T73164产 地：中国大陆
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T73161HadAB-IN-1；化合物 HadAB-IN-1HadAB-IN-1
HadAB-IN-1, a potent inhibitor of the HadAB enzyme complex, exhibits significant activity by restraining mycolic acid biosynthesis in Mycobacterium tuberculosis (Mtb), with an inhibitory concentration (IC 50) value of 0.03 μM. This compound is utilized in tuberculosis (TB) research.
价 格：￥电议型 号：T73161产 地：中国大陆
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T73151USP22-IN-1；化合物USP22-IN-1USP22-IN-1
USP22-IN-1 is a ubiquitin-specific peptidase 22 (USP22) inhibitor that can be used to treat proliferative diseases or cancer.
价 格：￥电议型 号：T73151产 地：中国大陆
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T73142FLT3-IN-18；化合物 FLT3-IN-18FLT3-IN-18
FLT3-IN-18, a potent and selective FLT3 inhibitor, exhibits an IC50 value of 0.003 μM. It effectively induces apoptosis and G1 phase cell cycle arrest, while inhibiting FLT3 and STAT5 phosphorylation. This compound holds potential for acute myeloid leukemia (AML) research.
价 格：￥电议型 号：T73142产 地：中国大陆
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T73136USP7-IN-10；化合物 USP7-IN-10USP7-IN-10
USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.
价 格：￥电议型 号：T73136产 地：中国大陆
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T73134EZH2-IN-14；化合物 EZH2-IN-14EZH2-IN-14
EZH2-IN-14 is a selective inhibitor of EZH2 (Histone Methyltransferase), demonstrating potent inhibition with an IC50 value of 12 nM. It specifically targets the methyltransferase activity of EZH2/PRC2, effectively reducing H3K27me3 levels. Moreover, EZH2-IN-14 exhibits more than 200-fold selectivity for EZH2 over the closely related H3K27 methyltransferase, EZH1.
价 格：￥电议型 号：T73134产 地：中国大陆
