您好，欢迎来到易推广！ 请登录 免费注册

上海陶术生物科技有限公司 主营产品：生物试剂,实验服务等

当前位置：易推广 > 上海陶术生物科技有限公司 > 产品展示

企业档案

会员类型：会员

已获得易推广信誉   等级评定
139成长值

(0 -40)基础信誉积累，可浏览访问

(41-90)良好信誉积累，可接洽商谈

(91+  )优质信誉积累，可持续信赖

易推广会员：5年

工商认证 【已认证】

最后认证时间：

注册号： 【已认证】

法人代表： 【已认证】

企业类型：生产商 【已认证】

注册资金：人民币万 【已认证】

产品数：86101

参观次数：3860936

手机网站：http://m.yituig.com/c135739/

旗舰版地址：http://tsbiochem.app17.com

自主品牌

自主品牌

已选条件

  • T61896hCAIX-IN-12；化合物 hCAIX-IN-12hCAIX-IN-12

    hCAIX-IN-12 is an effective hCAIX inhibitor, IC50 for CAIX and CAII is 0.74 and 10.78 μM , respectively. hCAIX-IN-12 inhibits cell proliferation and induces apoptosis. HCAIX-IN-12 can increase the generation of ROS. HCAIX-IN-12 has research potential in colorectal cancer (CRC).

    价 格：￥电议型 号：T61896产 地：中国大陆

  • T61893CSF1R-IN-12；化合物 CSF1R-IN-12CSF1R-IN-12

    CSF1R-IN-12 is an effective CSF1R inhibitor. CSF1R-IN-12 has research potential in cancer diseases.

    价 格：￥电议型 号：T61893产 地：中国大陆

  • T61888mTOR/HDAC6-IN-1；化合物 mTOR/HDAC6-IN-1mTOR/HDAC6-IN-1

    mTOR/HDAC6-IN-1 is an effective dual inhibitor of histone deacetylase (HDAC6) and mammalian rapamycin (mTOR). The IC50 values for HDAC6 and mTOR are 56 nM and 133.7 nM respectively. MTOR/HDAC6-IN-1 can significantly induce autophagy and apoptosis and inhibit migration. MTOR/HDAC6-IN-1 has potential in the study of triple negative breast cancer (TNBC).

    价 格：￥电议型 号：T61888产 地：中国大陆

  • T61887RIPK1-IN-13；化合物 RIPK1-IN-13RIPK1-IN-13

    RIPK1-IN-13 (Compound 8) is an effective RIPK1 inhibitor (IC50=1139 nM). By inhibiting RIPK1, RIPK1-IN-13 can block the activation of necrotic apoptosis pathway. RIPK1-IN-13 has research potential in inflammatory diseases.

    价 格：￥电议型 号：T61887产 地：中国大陆

  • T61886HBV-IN-16；化合物 HBV-IN-16HBV-IN-16

    HBV-IN-16 is a quinoline derivative, which has an effective inhibitory effect on covalent closed circular DNA (cccDNA). CccDNA is the template for viral RNA transcription and subsequent viral DNA generation. HBV-IN-16 has potential in the research of HBV infection.

    价 格：￥电议型 号：T61886产 地：中国大陆

  • T61873hCAIX/XII-IN-1；化合物 hCAIX/XII-IN-1hCAIX/XII-IN-1

    hCAIX/XII-IN-1, a potent inhibitor of both CAIX and CAXII, exhibits KI values of 0.48 μM for CAIX and 0.83 μM for CAXII, respectively. This compound demonstrates antiproliferative activity in vitro and induces apoptosis in MCF-7 cells [1].

    价 格：￥电议型 号：T61873产 地：中国大陆

  • T61872Trk-IN-10；化合物 Trk-IN-10Trk-IN-10

    Trk-IN-10 (Compound 14j) is a highly effective inhibitor of TRK, with an IC50 of 0.86 nM against TrkA and 6.92 nM against TrkA G595R. As an RTK, Trk plays a crucial role as a drug target in solid tumors. Trk-IN-10 (IC50 = 350 nM against ALK) demonstrates superior selectivity in inhibiting Trk, which has potential implications for toxicity reduction [1].

    价 格：￥电议型 号：T61872产 地：中国大陆

  • T61862PRMT5-IN-19；化合物 PRMT5-IN-19PRMT5-IN-19

    PRMT5-IN-19 (Compound 41) is a potent orally active PRMT5 inhibitor, exhibiting selectivity towards the SAM-binding pocket of PRMT5 with IC50 values of 23.9 nM (radioactive biochemical assay) and 47 nM (AlphaLISA assay). It effectively blocks methyltransferase activity and demonstrates high specificity against other PRMTs and PKMTs. PRMT5-IN-19 exerts anti-proliferative effects through the induction of apoptosis and holds potential in cancer-related research [1].

    价 格：￥电议型 号：T61862产 地：中国大陆

  • T61841SCD1-IN-1；化合物 SCD1-IN-1SCD1-IN-1

    SCD1-IN-1, a potent inhibitor of SCD1 (IC50: 5.8 nM), is valuable in dermatologic research [1].

    价 格：￥电议型 号：T61841产 地：中国大陆

  • T61831NS1-IN-1；化合物NS1-IN-1NS1-IN-1

    NS1-IN-1 is a potent NS1 inhibitor.NS1-IN-1 displays antiviral activity by inhibiting mTORC1 activity in a TSC1-TSC2-dependent manner.NS1-IN-1 reduces the level of viral proteins and contributes to the reduction of viral replication.

    价 格：￥电议型 号：T61831产 地：中国大陆

  • T61830MAO-B-IN-10；化合物 MAO-B-IN-10MAO-B-IN-10

    MAO-B-IN-10 (compound 4f) is a highly potent and selective inhibitor of MAO-B (monoamine oxidase-B). It effectively penetrates the blood-brain barrier and exhibits an IC50 of 5.3 μM. This compound demonstrates the ability to inhibit self-mediated Aβ (amyloid β) aggregation by 58.2% and disaggregate it by 43.3%. Thus, MAO-B-IN-10 holds promise for Alzheimer´s disease research [1].

    价 格：￥电议型 号：T61830产 地：中国大陆

  • T61821COX-2-IN-16；化合物 COX-2-IN-16COX-2-IN-16

    COX-2-IN-16 (compound 2b) is a potent, selective, and orally active inhibitor of cyclooxygenase-2 (COX-2) with an IC50 value of 102 μM. It effectively reduces nitric oxide (NO) production and demonstrates anti-inflammatory activity [1].

    价 格：￥电议型 号：T61821产 地：中国大陆

  • T61820Ar-V7-IN-1；化合物 Ar-V7-IN-1Ar-V7-IN-1

    Ar-V7-IN-1 is a highly potent inhibitor specifically targeting Ar-V7, a splice variant of the androgen receptor that exhibits hormone-independent behavior. Its development shows promise for researching various indications, notably cancers such as prostate cancer[1].

    价 格：￥电议型 号：T61820产 地：中国大陆

  • T61808ATR-IN-14；化合物 ATR-IN-14ATR-IN-14

    ATR-IN-14 (compound 1) is a powerful ATR kinase inhibitor that significantly inhibits ATR signaling pathways following CHKI protein phosphorylation, demonstrating a remarkable inhibition rate of 98.03% at 25 nM. Moreover, ATR-IN-14 exhibits notable anticancer efficacy in LoVo cells, displaying an IC50 value of 64 nM [1].

    价 格：￥电议型 号：T61808产 地：中国大陆

  • T61798PARP-1-IN-1；化合物 PARP-1-IN-1PARP-1-IN-1

    PARP-1-IN-1 is a highly selective and orally active inhibitor of the enzyme PARP-1, with an IC50 value of 0.96 nM. It exhibits excellent tolerance and demonstrates significant activity in a single dose in the MDA-MB-436 xenotransplantation model [1].

    价 格：￥电议型 号：T61798产 地：中国大陆

  • T61796MtTMPK-IN-1；化合物 MtTMPK-IN-1MtTMPK-IN-1

    MtTMPK-IN-1 (compound 3) is a highly effective inhibitor of Mycobacterium tuberculosis thymidylate kinase (Mt TMPK), exhibiting an IC50 value of 2.5 μM. It displays moderate to weak activity against Mtb H37Rv while demonstrating low cytotoxicity in human fibroblast cells MRC-5. MtTMPK-IN-1 is a valuable tool for tuberculosis research [1].

    价 格：￥电议型 号：T61796产 地：中国大陆

  • T61792HDAC6-IN-10；化合物 HDAC6-IN-10HDAC6-IN-10

    HDAC6-IN-10 is a potent and specific HDAC6 inhibitor, exhibiting an IC50 value of 0.73 nM. It demonstrates remarkable selectivity towards HDAC6, with a selectivity range of 144 to 10,941-fold over other HDAC isoforms. Furthermore, HDAC6-IN-10 exhibits notable anti-proliferative effects on multiple myeloma cells [1].

    价 格：￥电议型 号：T61792产 地：中国大陆

  • T61791BRD4-BD1/2-IN-1；化合物 BRD4-BD1/2-IN-1BRD4-BD1/2-IN-1

    BRD4-BD1/2-IN-1 is a highly effective inhibitor of BRD4, specifically targeting the BRD4 BD-1 and BRD4 BD-2 domains with IC 50 values of <100 nM each (US20150148375A1, compound 5) [1].

    价 格：￥电议型 号：T61791产 地：中国大陆

  • T61789IDO1-IN-14；化合物 IDO1-IN-14IDO1-IN-14

    IDO1-IN-14 (compound 4a) is a highly effective inhibitor of the IDO1 enzyme, exhibiting an IC50 value of 396.9 nM. Additionally, IDO1-IN-14 demonstrates excellent suppression of cellular IDO1 activity, as observed in HeLa cells with an EC50 value of 3393 nM [1].

    价 格：￥电议型 号：T61789产 地：中国大陆

  • T61784GlcN-6-P Synthase-IN-1；化合物 GlcN-6-P Synthase-IN-1GlcN-6-P Synthase-IN-1

    GlcN-6-P Synthase-IN-1 (Compound 4d) is a potent inhibitor of Glucosamine-6-phosphate (GlcN-6-P) synthase, with an IC50 of 3.47 μM. This compound demonstrates remarkable antimicrobial activity and exhibits excellent penetration in the central nervous system. Additionally, GlcN-6-P Synthase-IN-1 is capable of inhibiting cytochrome P450, specifically the CYP3A4 isoform [1].

    价 格：￥电议型 号：T61784产 地：中国大陆

162636465666768697071101下一页共101页

展台首页| 公司简介| 供应产品| 产品目录| 公司动态| 荣誉证书| 招聘信息| 技术中心| 联系我们| 会员管理

易推广  设计制作，未经允许翻录必究.Copyright(C) 2009 http://www.yituig.com, All rights reserved.

以上信息由企业自行提供，信息内容的真实性、准确性和合法性由相关企业负责，易推广对此不承担任何责任.   总访问量：3860936

中国彩虹热线

快速导航

返回顶部
在线咨询

提交